Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RFGOESLFDUAMGB
|
6.0 | IC50 | 4 | — | |
RTVPWYJBMHEYTA
|
6.0 | IC50 | 4 | — | |
SLUNFEBZDXASNJ
|
6.0 | IC50 | 4 | — | |
SVXHTPKAAXLDLX
|
6.0 | IC50 | 4 | — | |
SYPAMOJTLDNMQL
|
6.0 | IC50 | 4 | — | |
UDUFRUMXLFCNQN
|
6.0 | IC50 | 4 | — | |
UUGBZZQAHRXVBV
|
6.0 | IC50 | 4 | — | |
UZZOOCJSVGDZPS
|
6.0 | IC50 | 4 | — | |
VAEZIOUPBWPWKT
|
6.0 | IC50 | 4 | — | |
VLHPKUJISXSNFG
|
6.0 | IC50 | 4 | — | |
WHGYCNIXXDEKMI
|
6.0 | IC50 | 4 | — | |
WILCKYMTSIVKIZ
|
6.0 | IC50 | 4 | — | |
WLNHFWZZOOBEHX
|
6.0 | IC50 | 4 | — | |
WLSKWMBVRHXLLG
|
6.0 | IC50 | 4 | — | |
WREUMGOBADOOMR
|
6.0 | IC50 | 4 | — | |
WVWGMHSCWFAKFO
|
6.0 | IC50 | 4 | — | |
WWCJRXYIKMLMHV
|
6.0 | IC50 | 4 | — | |
WYNUQGLAIYDBRL
|
6.0 | IC50 | 4 | — | |
XAWMWRRMUXYKPC
|
6.0 | IC50 | 4 | — | |
XDDFKFMQTWAHQW
|
6.0 | IC50 | 4 | — | |
XOEWAGGFKMWDPJ
|
6.0 | IC50 | 4 | — | |
YASUGMSGTIVYCC
|
6.0 | IC50 | 4 | — | |
YAYMVYXCAZWMFA
|
6.0 | IC50 | 4 | — | |
ZRJGAZHGDXMXNT
|
6.0 | IC50 | 4 | — |