Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RQHOVOFQMVYWSJ
|
6.1 | IC50 | 3 | — | |
BEJPKJRTOYTNEK
|
6.1 | IC50 | 3 | — | |
QGVSLEINXMWQMT
|
6.0 | IC50 | 4 | — | |
AFRYLLNYYFRUKZ
|
6.0 | IC50 | 4 | — | |
AIDMBUXHQJQJMB
|
6.0 | IC50 | 4 | — | |
AVIBHWXBXPFMLQ
|
6.0 | IC50 | 4 | — | |
BOCXGAVHERNIED
|
6.0 | IC50 | 4 | — | |
BOGRKBZCGGVGGS
|
6.0 | IC50 | 4 | — | |
BVSMEZQQQTUAMN
|
6.0 | IC50 | 4 | — | |
CBHNHZXDESJXQZ
|
6.0 | IC50 | 4 | — | |
CKCBDRGQGSQRFN
|
6.0 | IC50 | 4 | — | |
CWAXXGRNESDIFD
|
6.0 | IC50 | 4 | — | |
DFBBARPBDNOHIG
|
6.0 | IC50 | 4 | — | |
DRJCGVYRZOBJOV
|
6.0 | IC50 | 4 | — | |
FMLYGCPVSHVBGL
|
6.0 | IC50 | 4 | — | |
FMTIOPPCYVSTGQ
|
6.0 | IC50 | 4 | — | |
FOHLYNYTSUJQTP
|
6.0 | IC50 | 4 | — | |
FQMNWBLEFIAYPW
|
6.0 | IC50 | 4 | — | |
GHNVNCXYLHYQDO
|
6.0 | IC50 | 4 | — | |
GKSNEZLHIIZEGL
|
6.0 | IC50 | 4 | — | |
GXNHMFDKLVMBBF
|
6.0 | IC50 | 4 | — | |
HGWPYDZYRWUXAC
|
6.0 | IC50 | 4 | — | |
HXEZLTWOXMXCJJ
|
6.0 | IC50 | 4 | — | |
IEPMJKSTICKITB
|
6.0 | IC50 | 4 | — | |
JBXCZTFOQMGTBA
|
6.0 | IC50 | 4 | — | |
JCMGJBTYTUCSSM
|
6.0 | IC50 | 4 | — | |
JLWRTIPIGXDNEG
|
6.0 | IC50 | 4 | — | |
JQHAKNWHEFDSNQ
|
6.0 | IC50 | 4 | — | |
JQHNJRAABZZPFN
|
6.0 | IC50 | 4 | — | |
JXGCDBJFNMMLNB
|
6.0 | IC50 | 4 | — | |
JZKWCVYCWBMBFY
|
6.0 | IC50 | 4 | — | |
JZQRWFCPYXTEEC
|
6.0 | IC50 | 4 | — | |
KHTIYNJMMLQJRX
|
6.0 | IC50 | 4 | — | |
KMWHNYZBANTQFA
|
6.0 | IC50 | 4 | — | |
KZGYMLHJMGQXOM
|
6.0 | IC50 | 4 | — | |
LBPOGQUABVQXPM
|
6.0 | IC50 | 4 | — | |
LMKXJIKIUSIWSP
|
6.0 | IC50 | 4 | — | |
LSBCJXWWDZEWRF
|
6.0 | IC50 | 4 | — | |
LVNJKOIEYNEOMZ
|
6.0 | IC50 | 4 | — | |
MJTMTQQRDNWPGK
|
6.0 | IC50 | 4 | — | |
MMLLULKUDKWCNR
|
6.0 | IC50 | 4 | — | |
NPZRDYRAAKIHPY
|
6.0 | IC50 | 4 | — | |
OINIDTBTTIYZIO
|
6.0 | IC50 | 4 | — | |
PUHWWAJTHDKCGR
|
6.0 | IC50 | 4 | — | |
PWDYOVIZDCYFRZ
|
6.0 | IC50 | 4 | — | |
PXUOKRBBSRTUNE
|
6.0 | IC50 | 4 | — | |
PZPMTBAIXNMBME
|
6.0 | IC50 | 4 | — | |
QQMKDSHSGYQMOV
|
6.0 | IC50 | 4 | — | |
QXCUSMAHYXWCOF
|
6.0 | IC50 | 4 | — | |
RECOPQDOXFPBNE
|
6.0 | IC50 | 4 | — |