Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.3 | IC50 | 408 | — | |
CECDQIYLZLGLFB
|
8.5 | IC50 | 2 | — | |
FDOLTFPOFUHZNO
|
8.5 | IC50 | 2 | — | |
FGTWUFDOPUTMFJ
|
8.5 | IC50 | 2 | — | |
QCTYBINXRYFEKA
|
8.5 | IC50 | 2 | — | |
QZHDUIFHCNLGNF
|
8.5 | IC50 | 2 | — | |
SEKVOZNRIOJKIM
|
8.5 | IC50 | 2 | — | |
UVOKTZOYQUAPBT
|
8.5 | IC50 | 2 | — | |
VPEYFYPTRQBQBA
|
8.5 | IC50 | 2 | — | |
WBTFLXDXOVVNOA
|
8.5 | IC50 | 2 | — | |
WVXGQODAPLIYFL
|
8.5 | IC50 | 2 | — | |
XNQCEAYNRGEWSL
|
8.5 | IC50 | 2 | — | |
YANYTYPXWFMHEC
|
8.5 | IC50 | 2 | — | |
YDLPFGWWTYFQLG
|
8.5 | IC50 | 2 | — | |
AFZAEHYINXKGIX
|
8.4 | IC50 | 2 | — | |
AYTOJFMWRQGYCF
|
8.4 | IC50 | 2 | — | |
BCIZDBFLZAGDOJ
|
8.4 | IC50 | 2 | — | |
BUTPPJYHAKFGSS
|
8.4 | IC50 | 2 | — | |
CKFGGNAQXLOYTI
|
8.4 | IC50 | 2 | — | |
CZAKHJFTIYBXDG
|
8.4 | IC50 | 2 | — | |
DMRFRHLBWMTTBS
|
8.4 | IC50 | 2 | — | |
DXLWIZJIQBYXMG
|
8.4 | IC50 | 2 | — | |
GEEAWGMCDJTFDL
|
8.4 | IC50 | 2 | — | |
IPRDTYTVGQVNPC
|
8.4 | IC50 | 2 | — | |
IXSFFXAAURBUCO
|
8.4 | IC50 | 2 | — | |
JBOUJRQXBKCBNJ
|
8.4 | IC50 | 2 | — | |
MPCBDAXTWLZHRP
|
8.4 | IC50 | 2 | — | |
NCMNSDQGHJLYTB
|
8.4 | IC50 | 3 | — | |
OSVUGUHRKMMBSE
|
8.4 | Kd | 170 | — | |
PJBJZXQMMLTSPW
|
8.4 | IC50 | 2 | — | |
RXEHIULELGCSKA
|
8.4 | IC50 | 2 | — | |
SDYHYNUKUWSPFA
|
8.4 | IC50 | 2 | — | |
UKZUEAUSMNCXCT
|
8.4 | IC50 | 2 | — | |
WYGPZNHUVVHVKK
|
8.4 | IC50 | 2 | — | |
XDLRILQJNLAQLU
|
8.4 | IC50 | 2 | — | |
ADUOVQPGZNRALP
|
8.3 | IC50 | 2 | — | |
BADAASATSUKKRC
|
8.3 | IC50 | 2 | — | |
BNSMNQFWANUEIK
|
8.3 | IC50 | 2 | — | |
GDMZIUSWFQWRIG
|
8.3 | IC50 | 2 | — | |
GXBGRQPGTWTRDX
|
8.3 | IC50 | 2 | — | |
GZZMQXYSLCBPEA
|
8.3 | IC50 | 2 | — | |
JHDVCYUKJXSYAA
|
8.3 | IC50 | 2 | — | |
KLDQUPYWEFWFQK
|
8.3 | IC50 | 2 | — | |
NUIADYLLUQJNJC
|
8.3 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
8.3 | Kd | 200 | — | |
PBKHUXFKXFHMMJ
|
8.3 | IC50 | 2 | — | |
PBOGEDJQULJRGL
|
8.3 | IC50 | 2 | — | |
PNECHCFDYAQPCJ
|
8.3 | IC50 | 2 | — | |
QLPHOXTXAKOFMU
|
8.3 | IC50 | 2 | — | |
QMVPFGNVCUNBET
|
8.3 | IC50 | 2 | — |