Target Details
| UniProt AC | Q15078 |
|---|---|
| Gene Symbol | CDK5R1 |
| Protein Name | Cyclin-dependent kinase 5 activator 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03261 (CDK5_activator) |
Summary
- Multi-target molecules 891
- Clinical molecules 54
- Avg pChEMBL 6.92
KEGG Pathways (3)
Active Molecules (891)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KIHCZOJSOYPCCE
|
7.1 | IC50 | 2 | — | |
PMXCMJLOPOFPBT
|
7.1 | IC50 | 17 | Yes | |
ZPKXDHHDZZKMKI
|
7.1 | IC50 | 6 | — | |
JEWCMAYLACWOQD
|
7.1 | IC50 | 2 | — | |
YPSCKJWJIXZMSC
|
7.1 | IC50 | 15 | — | |
ZUCAWWSJZRVUAX
|
7.1 | Ki | 11 | — | |
BGNDQDYZQSRSAU
|
7.1 | IC50 | 3 | — | |
BGQVVTJSMBYUHC
|
7.1 | IC50 | 2 | — | |
BGQVVTJSMBYUHC
|
7.1 | IC50 | 2 | — | |
GLDKGDSJAPIZTI
|
7.1 | IC50 | 2 | — | |
KVVMSGAISWJACO
|
7.1 | IC50 | 3 | — | |
MAUHUPWBMYAXPZ
|
7.1 | IC50 | 2 | — | |
NOOMEBXFKHIBIE
|
7.1 | IC50 | 2 | — | |
DDLZLOKCJHBUHD
|
7.1 | IC50 | 23 | — | |
HGRMYMRCAGWXEQ
|
7.1 | IC50 | 6 | — | |
OLOJSTRISMGUEK
|
7.1 | IC50 | 5 | — | |
PFDVIMSWMQLRQB
|
7.1 | IC50 | 2 | — | |
ZPHBEDTYTQWLFC
|
7.1 | IC50 | 13 | — | |
NXSJMRCTGYTSTK
|
7.1 | Kd | 200 | — | |
AREWHVALAPEARZ
|
7.0 | IC50 | 4 | — | |
IWXIAMLCFOOOMV
|
7.0 | IC50 | 8 | Yes | |
PRRNEKPNFWMEPT
|
7.0 | IC50 | 2 | — | |
UNLGUYJWTWLABD
|
7.0 | IC50 | 2 | — | |
VMSMVRDDPGJMQF
|
7.0 | IC50 | 5 | — | |
CEIJSVLEARLWRF
|
7.0 | IC50 | 13 | — | |
CQVJGFKTRSGJHB
|
7.0 | Ki | 11 | — | |
GJTRIRZIYRVGHG
|
7.0 | IC50 | 4 | — | |
QNWXRLPZIFMTBK
|
7.0 | IC50 | 12 | — | |
SVPUOZWGAJVQMQ
|
7.0 | IC50 | 2 | — | |
YWZXVOUKTPVGKU
|
7.0 | IC50 | 2 | — | |
KGMVZSJAPXYTKH
|
7.0 | IC50 | 23 | — | |
DMFMPEWLXMKYKK
|
7.0 | IC50 | 4 | — | |
FQCPPVRJPILDIK
|
7.0 | IC50 | 12 | — | |
HBDSHCUSXQATPO
|
7.0 | IC50 | 14 | Yes | |
HKECWLZKPZHUND
|
7.0 | IC50 | 8 | — | |
HOQNHSNBIIJJBO
|
7.0 | IC50 | 7 | — | |
HWUAECSPBXTMLX
|
7.0 | IC50 | 2 | — | |
JSJVSQMHVJPNON
|
7.0 | IC50 | 5 | — | |
PBTNYNHOVGFGNO
|
7.0 | IC50 | 2 | — | |
TVUWQDLBEOZVOU
|
7.0 | IC50 | 41 | — | |
ZLNVBIGZYRPQKY
|
7.0 | IC50 | 15 | — | |
HLUQDCJXKVVBRH
|
7.0 | IC50 | 2 | — | |
BKLVJGBLXVWFCJ
|
7.0 | IC50 | 3 | Yes | |
CIDXXRSLUUUBDG
|
7.0 | IC50 | 2 | — | |
FHDFIUFWMGMGTR
|
7.0 | IC50 | 5 | — | |
ISYFANQBAGVSNZ
|
7.0 | IC50 | 2 | — | |
JOKSIWLEZWYCLI
|
7.0 | IC50 | 2 | — | |
XOXWOPNBJDVSJP
|
7.0 | Ki | 8 | — | |
ZSSHCAVAAPDLII
|
7.0 | IC50 | 5 | — | |
JYRJOQGKGMHTOO
|
7.0 | IC50 | 9 | — |