Target Details
| UniProt AC | Q15078 |
|---|---|
| Gene Symbol | CDK5R1 |
| Protein Name | Cyclin-dependent kinase 5 activator 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03261 (CDK5_activator) |
Summary
- Multi-target molecules 891
- Clinical molecules 54
- Avg pChEMBL 6.92
KEGG Pathways (3)
Active Molecules (891)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XNKBKFNLOYVTSF
|
7.2 | IC50 | 11 | — | |
CLTHCEMHDXFICR
|
7.2 | IC50 | 2 | — | |
AYSFEKIVJXIJTM
|
7.2 | IC50 | 8 | — | |
BOPIEFLHGAQWGB
|
7.2 | IC50 | 3 | — | |
HLSGDZZAUXGGFJ
|
7.2 | Ki | 4 | — | |
LQYHWFFRRIMAPW
|
7.2 | IC50 | 2 | — | |
RSPXQCXRWMXEAA
|
7.2 | IC50 | 2 | — | |
SBNNOXYSSSCMJX
|
7.2 | IC50 | 6 | — | |
SJJOSGWHLXBKSU
|
7.2 | IC50 | 2 | — | |
TUMYZJPVQGGVEN
|
7.2 | IC50 | 7 | — | |
XCRSLBLUJPTVDN
|
7.2 | IC50 | 3 | — | |
GRMBHDGZBLMPSZ
|
7.2 | IC50 | 2 | — | |
JBTRAENEEJNXFX
|
7.2 | IC50 | 2 | — | |
KCGZOQMFGRRYKH
|
7.2 | IC50 | 3 | — | |
KKNOSXFGCMVMNP
|
7.2 | IC50 | 2 | — | |
MAIBFWJHQLEUMH
|
7.2 | IC50 | 2 | — | |
NGFGTMFVWSDFPS
|
7.2 | IC50 | 32 | — | |
WMIYIBXBFBOKCT
|
7.2 | IC50 | 3 | — | |
WMIYIBXBFBOKCT
|
7.2 | IC50 | 6 | — | |
YOOLJWCJXSFKSE
|
7.2 | IC50 | 2 | — | |
ZJKDYTFNXUBLEQ
|
7.2 | IC50 | 15 | — | |
HQUWRDCCNSLORW
|
7.2 | IC50 | 2 | — | |
FRLPUUILIGCJSG
|
7.2 | IC50 | 2 | — | |
IHBOEHLUIBMBMY
|
7.2 | IC50 | 7 | Yes | |
MOFKVWKHBJPHSX
|
7.2 | IC50 | 2 | — | |
NUBBIJVOSXWZTF
|
7.2 | IC50 | 13 | — | |
QYCAOWUXVAQWNK
|
7.2 | IC50 | 2 | — | |
SHHLIGVBIWQSRR
|
7.2 | IC50 | 4 | — | |
UAOIPNOTWOYAMU
|
7.2 | IC50 | 11 | Yes | |
XGWCLSYLELRSQN
|
7.2 | IC50 | 2 | — | |
YIAFFFACXVWBIZ
|
7.2 | IC50 | 4 | — | |
ZHRBVPKKEHKSFH
|
7.2 | IC50 | 4 | — | |
HCRMONBJZIFRIR
|
7.2 | IC50 | 4 | — | |
LNLSVTCWVQLNIY
|
7.2 | IC50 | 2 | — | |
WROPYEAREMSHKX
|
7.2 | IC50 | 2 | — | |
XVNXLMMYWHJXME
|
7.2 | IC50 | 2 | — | |
BRQIEVOYMRUXNP
|
7.2 | IC50 | 7 | — | |
CFVOEIRDSYTLGT
|
7.2 | IC50 | 2 | — | |
GYEMABRPKRSBJU
|
7.2 | IC50 | 2 | — | |
SQUNOCMDMIQIQK
|
7.2 | IC50 | 10 | — | |
ULWKEYMEZWWCRY
|
7.2 | Ki | 5 | — | |
CXMKIWPGGSLHRE
|
7.2 | IC50 | 15 | — | |
KGLQVHSLHDKNTQ
|
7.2 | IC50 | 4 | — | |
CIBYULXUPNERCM
|
7.1 | IC50 | 2 | — | |
NKSJUACUARPPLH
|
7.1 | IC50 | 13 | — | |
QIYYNXDEQKBHEH
|
7.1 | IC50 | 5 | — | |
SFDWUKJFXSWJPJ
|
7.1 | IC50 | 2 | — | |
WKEZGEHTYROLRA
|
7.1 | IC50 | 2 | — | |
JFEXQCAPNBAVHH
|
7.1 | IC50 | 2 | — | |
JFEXQCAPNBAVHH
|
7.1 | IC50 | 2 | — |