Target Details
UniProt ACQ15078
Gene SymbolCDK5R1
Protein NameCyclin-dependent kinase 5 activator 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF03261 (CDK5_activator)
Summary
  • Multi-target molecules 891
  • Clinical molecules 54
  • Avg pChEMBL 6.92
Top Co-occurrence Targets
Active Molecules (891)
InChIKey pChEMBL Type Targets Clinical
XNKBKFNLOYVTSF 7.2 IC50 11
CLTHCEMHDXFICR 7.2 IC50 2
AYSFEKIVJXIJTM 7.2 IC50 8
BOPIEFLHGAQWGB 7.2 IC50 3
HLSGDZZAUXGGFJ 7.2 Ki 4
LQYHWFFRRIMAPW 7.2 IC50 2
RSPXQCXRWMXEAA 7.2 IC50 2
SBNNOXYSSSCMJX 7.2 IC50 6
SJJOSGWHLXBKSU 7.2 IC50 2
TUMYZJPVQGGVEN 7.2 IC50 7
XCRSLBLUJPTVDN 7.2 IC50 3
GRMBHDGZBLMPSZ 7.2 IC50 2
JBTRAENEEJNXFX 7.2 IC50 2
KCGZOQMFGRRYKH 7.2 IC50 3
KKNOSXFGCMVMNP 7.2 IC50 2
MAIBFWJHQLEUMH 7.2 IC50 2
NGFGTMFVWSDFPS 7.2 IC50 32
WMIYIBXBFBOKCT 7.2 IC50 3
WMIYIBXBFBOKCT 7.2 IC50 6
YOOLJWCJXSFKSE 7.2 IC50 2
ZJKDYTFNXUBLEQ 7.2 IC50 15
HQUWRDCCNSLORW 7.2 IC50 2
FRLPUUILIGCJSG 7.2 IC50 2
IHBOEHLUIBMBMY 7.2 IC50 7 Yes
MOFKVWKHBJPHSX 7.2 IC50 2
NUBBIJVOSXWZTF 7.2 IC50 13
QYCAOWUXVAQWNK 7.2 IC50 2
SHHLIGVBIWQSRR 7.2 IC50 4
UAOIPNOTWOYAMU 7.2 IC50 11 Yes
XGWCLSYLELRSQN 7.2 IC50 2
YIAFFFACXVWBIZ 7.2 IC50 4
ZHRBVPKKEHKSFH 7.2 IC50 4
HCRMONBJZIFRIR 7.2 IC50 4
LNLSVTCWVQLNIY 7.2 IC50 2
WROPYEAREMSHKX 7.2 IC50 2
XVNXLMMYWHJXME 7.2 IC50 2
BRQIEVOYMRUXNP 7.2 IC50 7
CFVOEIRDSYTLGT 7.2 IC50 2
GYEMABRPKRSBJU 7.2 IC50 2
SQUNOCMDMIQIQK 7.2 IC50 10
ULWKEYMEZWWCRY 7.2 Ki 5
CXMKIWPGGSLHRE 7.2 IC50 15
KGLQVHSLHDKNTQ 7.2 IC50 4
CIBYULXUPNERCM 7.1 IC50 2
NKSJUACUARPPLH 7.1 IC50 13
QIYYNXDEQKBHEH 7.1 IC50 5
SFDWUKJFXSWJPJ 7.1 IC50 2
WKEZGEHTYROLRA 7.1 IC50 2
JFEXQCAPNBAVHH 7.1 IC50 2
JFEXQCAPNBAVHH 7.1 IC50 2
2D structure