Target Details
| UniProt AC | Q15078 |
|---|---|
| Gene Symbol | CDK5R1 |
| Protein Name | Cyclin-dependent kinase 5 activator 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03261 (CDK5_activator) |
Summary
- Multi-target molecules 891
- Clinical molecules 54
- Avg pChEMBL 6.92
KEGG Pathways (3)
Active Molecules (891)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PDAAWAZSKXRPAS
|
7.4 | IC50 | 2 | — | |
DWDSNANBEINKNN
|
7.4 | IC50 | 4 | — | |
BIDYUGXUCHBVIV
|
7.4 | IC50 | 2 | — | |
HKOGEZCYHMAXBA
|
7.4 | IC50 | 2 | — | |
OLUKILHGKRVDCT
|
7.4 | IC50 | 44 | Yes | |
RMEWJCSHDSUJKS
|
7.4 | IC50 | 2 | — | |
DHPKYHMTJHTQKB
|
7.4 | IC50 | 2 | — | |
HFEVNTGRPXCJIM
|
7.4 | IC50 | 6 | — | |
CNNQBAXDFGTALM
|
7.4 | IC50 | 5 | — | |
CNNQBAXDFGTALM
|
7.4 | IC50 | 2 | — | |
GPSDJCPWZFYLRU
|
7.4 | IC50 | 2 | — | |
QYNVMKNYPFKRBL
|
7.4 | Ki | 9 | — | |
QZTJCAGUOSLOOZ
|
7.4 | IC50 | 2 | — | |
SBNNOXYSSSCMJX
|
7.4 | IC50 | 6 | — | |
UUFIEDRPFIIXAY
|
7.4 | Ki | 6 | — | |
ZPKXDHHDZZKMKI
|
7.4 | IC50 | 6 | — | |
BHGNYQXAUNNTRE
|
7.4 | IC50 | 2 | — | |
OSZOLMOXJMNVGS
|
7.4 | IC50 | 4 | — | |
FEUVVQAFOCJYBF
|
7.4 | IC50 | 2 | — | |
JVLUKLANRWXEHV
|
7.4 | IC50 | 2 | — | |
KEUUTBKQXWXFLI
|
7.4 | IC50 | 5 | — | |
LBVIZFWUIQSZHP
|
7.4 | IC50 | 10 | — | |
URMALQKFRQFSGH
|
7.4 | IC50 | 2 | — | |
CQZDWCOZFXQUFP
|
7.3 | IC50 | 2 | — | |
DBDLWYCQSVIKRY
|
7.3 | IC50 | 2 | — | |
KAMWROHYXYCDLF
|
7.3 | IC50 | 2 | — | |
IRLVKSQKZPUCOP
|
7.3 | IC50 | 2 | — | |
LBPVERPKZZCMIU
|
7.3 | IC50 | 2 | — | |
NGLJEWVPKWMIAJ
|
7.3 | IC50 | 5 | — | |
SMWJYKRUKGMKJV
|
7.3 | IC50 | 11 | — | |
ULNGKSGQVVQHJF
|
7.3 | IC50 | 2 | — | |
FSEJNURQBJZNAM
|
7.3 | IC50 | 2 | — | |
JYGNOLIKBUTZNC
|
7.3 | IC50 | 8 | Yes | |
NTHMDBBWWNTVAZ
|
7.3 | IC50 | 5 | — | |
PRJNNPMIUGYOST
|
7.3 | IC50 | 14 | — | |
RAFWSIQGGUBJOQ
|
7.3 | IC50 | 2 | — | |
SVBJNUDKKXGVHI
|
7.3 | IC50 | 6 | — | |
WAWDNROIUWNCQG
|
7.3 | IC50 | 2 | — | |
WROPYEAREMSHKX
|
7.3 | IC50 | 2 | — | |
GNTSKAUZBDGNGK
|
7.3 | IC50 | 6 | — | |
IPSJLLWTAZLENF
|
7.3 | IC50 | 2 | — | |
RXGOWNXDRJHZDW
|
7.3 | IC50 | 2 | — | |
DPFVGQNGSOMJSY
|
7.3 | IC50 | 2 | — | |
JLKHGQLTVZHANW
|
7.3 | IC50 | 2 | — | |
VCEUNJCUQFBRBD
|
7.3 | IC50 | 2 | — | |
CQGFDYLOZSKCBQ
|
7.3 | IC50 | 2 | — | |
ZITKTAJHKVYGTC
|
7.2 | IC50 | 4 | — | |
ZITKTAJHKVYGTC
|
7.2 | IC50 | 7 | — | |
HONCRTYDCHPQOK
|
7.2 | IC50 | 2 | — | |
WRPCQNMNBWSPBJ
|
7.2 | IC50 | 2 | — |