Target Details
| UniProt AC | Q15078 |
|---|---|
| Gene Symbol | CDK5R1 |
| Protein Name | Cyclin-dependent kinase 5 activator 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03261 (CDK5_activator) |
Summary
- Multi-target molecules 891
- Clinical molecules 54
- Avg pChEMBL 6.92
KEGG Pathways (3)
Active Molecules (891)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IORBEYRNTKWGRM
|
7.6 | IC50 | 4 | — | |
MZWFSHNLGOBBSZ
|
7.6 | IC50 | 2 | — | |
POCZBHBFCIWCCV
|
7.6 | IC50 | 5 | — | |
VCTLOEWZYIGVBO
|
7.6 | IC50 | 12 | — | |
VMSMVRDDPGJMQF
|
7.6 | IC50 | 6 | — | |
BZAMUGWDAXKCEU
|
7.6 | IC50 | 2 | — | |
UTBSBSOBZHXMHI
|
7.6 | IC50 | 15 | Yes | |
ATBAETXFFCOZOY
|
7.6 | IC50 | 39 | — | |
HHZHUPXWPPYGEU
|
7.6 | IC50 | 4 | — | |
YZSCPLGKKMSBMV
|
7.6 | IC50 | 10 | — | |
DSEWGOFKGFEZPE
|
7.5 | IC50 | 2 | — | |
IZOFFSRJFXHBHQ
|
7.5 | IC50 | 2 | — | |
LDLLFYVEDBJIIM
|
7.5 | IC50 | 2 | — | |
TYNCGTPANDPODX
|
7.5 | IC50 | 4 | — | |
DENJPOISBSHUGX
|
7.5 | IC50 | 2 | — | |
PGDIYOJSLLUWMQ
|
7.5 | Ki | 4 | — | |
HHZHUPXWPPYGEU
|
7.5 | IC50 | 4 | — | |
MKNYSPZGSGBELV
|
7.5 | IC50 | 2 | — | |
NSEKTECTEUZVNV
|
7.5 | IC50 | 4 | — | |
PHZDWQYTFQOSSZ
|
7.5 | IC50 | 15 | — | |
SLKSRHOPMDATBX
|
7.5 | IC50 | 5 | — | |
SLKSRHOPMDATBX
|
7.5 | IC50 | 2 | — | |
UEFVCKVWJQJSDH
|
7.5 | IC50 | 2 | — | |
XHJMMMPXTUEBMQ
|
7.5 | IC50 | 4 | — | |
JFHNULPYENHDTR
|
7.5 | IC50 | 2 | — | |
TVQIAQPBIDLYOL
|
7.5 | IC50 | 4 | — | |
ZOPGCNRZFZPRGB
|
7.5 | Ki | 9 | — | |
OYPIIVNTYVSCNV
|
7.5 | IC50 | 4 | — | |
VGGPBVXGHSIMPS
|
7.5 | IC50 | 4 | — | |
KHYRHFAJCMYVAX
|
7.5 | IC50 | 2 | — | |
KVZRUJJMBHTJLY
|
7.5 | IC50 | 2 | — | |
PPSLREGORUQEEL
|
7.5 | IC50 | 2 | — | |
SHBOZSJPVRMXBA
|
7.5 | IC50 | 7 | — | |
TVARIYLSKVWCHN
|
7.5 | Ki | 11 | — | |
DBKUHLGRJZFKQS
|
7.5 | IC50 | 5 | — | |
FULPDCCIDPUWGS
|
7.5 | IC50 | 4 | — | |
LNGGMJFRIWMXLS
|
7.5 | IC50 | 2 | — | |
FDJQQPZQIBTWLE
|
7.5 | IC50 | 4 | — | |
PWWHQERJKXLERO
|
7.5 | IC50 | 2 | — | |
LLFOBMRPWNABCB
|
7.5 | IC50 | 11 | — | |
BUVUGYVWVBFUMI
|
7.4 | Ki | 11 | — | |
BYFFLCLXJMXMTM
|
7.4 | IC50 | 2 | — | |
FJINXQDJHXTMEL
|
7.4 | Ki | 9 | — | |
ATBAETXFFCOZOY
|
7.4 | IC50 | 10 | — | |
FYBVVRIGUJAAOT
|
7.4 | IC50 | 2 | — | |
RPYUTGQONYNCSI
|
7.4 | IC50 | 4 | — | |
FQFGDUPFMGYOMB
|
7.4 | IC50 | 6 | — | |
HCEVZIBGQRWFCG
|
7.4 | IC50 | 9 | — | |
HEPOPUWWRFFLLL
|
7.4 | IC50 | 2 | — | |
KMWYBWMCMDBJGT
|
7.4 | IC50 | 2 | — |