Target Details
| UniProt AC | Q15078 |
|---|---|
| Gene Symbol | CDK5R1 |
| Protein Name | Cyclin-dependent kinase 5 activator 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03261 (CDK5_activator) |
Summary
- Multi-target molecules 891
- Clinical molecules 54
- Avg pChEMBL 6.92
KEGG Pathways (3)
Active Molecules (891)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.0 | IC50 | 49 | Yes | |
IVPOEQUCSQIXKZ
|
8.0 | IC50 | 2 | — | |
NYCKILAUMKSIPT
|
8.0 | IC50 | 2 | — | |
ONPNTUDUPZVQGU
|
8.0 | IC50 | 2 | — | |
RWSCYFXGWJPUQX
|
8.0 | IC50 | 15 | — | |
UCAUIDINMHWADR
|
8.0 | IC50 | 4 | — | |
BBSNLVGUSKQSBU
|
7.9 | IC50 | 2 | — | |
BBSNLVGUSKQSBU
|
7.9 | IC50 | 2 | — | |
FKAJEPVSQITQLJ
|
7.9 | IC50 | 15 | — | |
TVKHEKZVCHMORX
|
7.9 | IC50 | 2 | — | |
TVKHEKZVCHMORX
|
7.9 | IC50 | 3 | — | |
ORKSQVXJLGIROJ
|
7.9 | IC50 | 4 | — | |
SYKKXAMILDNUNO
|
7.9 | IC50 | 4 | — | |
DIWRYQKRDLUVMY
|
7.8 | IC50 | 2 | — | |
KGJVKYSVVOQPDL
|
7.8 | IC50 | 13 | — | |
NPXTWLXCVUMFMN
|
7.8 | IC50 | 2 | — | |
FLIVKVQMXOAQAK
|
7.8 | IC50 | 15 | — | |
NBSJZWFDNFWQDN
|
7.8 | IC50 | 29 | — | |
PCQPAKMJSYGXRE
|
7.8 | IC50 | 16 | — | |
VSFIYAYRTKMILQ
|
7.8 | IC50 | 2 | — | |
DSHAIQLEQCKJIR
|
7.8 | IC50 | 7 | — | |
DVBHEDLDLJERFO
|
7.8 | Ki | 9 | — | |
NFTJDXGFOUFNKG
|
7.8 | IC50 | 16 | — | |
PIMQWRZWLQKKBJ
|
7.8 | IC50 | 36 | — | |
QHNBDDABNDUESC
|
7.8 | IC50 | 3 | — | |
FKAJEPVSQITQLJ
|
7.8 | IC50 | 15 | — | |
SVBJNUDKKXGVHI
|
7.8 | IC50 | 5 | — | |
GANPMWWREYHGFT
|
7.7 | IC50 | 2 | — | |
MNKJDIFJOOLBQY
|
7.7 | IC50 | 3 | Yes | |
OVPNQJVDAFNBDN
|
7.7 | IC50 | 44 | Yes | |
WROPYEAREMSHKX
|
7.7 | IC50 | 2 | — | |
FZLZLIAOYSKHJC
|
7.7 | Ki | 11 | — | |
QNABDSWBQJKBHK
|
7.7 | IC50 | 45 | — | |
UVKLAINVJNUJNX
|
7.7 | IC50 | 10 | — | |
BOLOCLITWRGHFA
|
7.7 | IC50 | 6 | — | |
VSLRVJBKRNJMHM
|
7.7 | IC50 | 2 | — | |
WCCYEJYTLNWYCC
|
7.7 | IC50 | 9 | — | |
ZJVHTWKAZJOGEG
|
7.7 | IC50 | 3 | — | |
DLPIYBKBHMZCJI
|
7.7 | IC50 | 12 | — | |
KYRQRRGDKAIFMA
|
7.7 | IC50 | 7 | — | |
NCBDOQFSGNRAHL
|
7.7 | IC50 | 6 | — | |
ASRWRMWLFZMROI
|
7.7 | IC50 | 6 | — | |
QNUKRWAIZMBVCU
|
7.7 | IC50 | 17 | Yes | |
ABTODZKWEKKTIC
|
7.6 | IC50 | 2 | — | |
DTNFOGMAASDEQI
|
7.6 | IC50 | 5 | — | |
LVELIXLMLUGJEH
|
7.6 | IC50 | 4 | — | |
LRJIEZPKWFBSEJ
|
7.6 | IC50 | 6 | — | |
PTAPBELLLOUDLL
|
7.6 | IC50 | 2 | — | |
QTHCAAFKVUWAFI
|
7.6 | IC50 | 23 | — | |
GFPGWHOCRYTVLL
|
7.6 | IC50 | 3 | — |