Target Details
| UniProt AC | Q15078 |
|---|---|
| Gene Symbol | CDK5R1 |
| Protein Name | Cyclin-dependent kinase 5 activator 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03261 (CDK5_activator) |
Summary
- Multi-target molecules 891
- Clinical molecules 54
- Avg pChEMBL 6.92
KEGG Pathways (3)
Active Molecules (891)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BXQKMGAINGBZAW
|
8.5 | IC50 | 11 | — | |
DYHPOLTXTOPHPD
|
8.5 | IC50 | 2 | — | |
DZKMAWNYSJECKX
|
8.5 | IC50 | 12 | — | |
FGNHJXSBQQICEW
|
8.4 | Ki | 7 | — | |
IEGUVVCSOPRFMZ
|
8.4 | IC50 | 4 | — | |
HUHQPIYUPMEDGV
|
8.4 | IC50 | 2 | — | |
WADWOQCKXASRGQ
|
8.4 | IC50 | 4 | — | |
VASFNXBXECJRSY
|
8.4 | IC50 | 15 | — | |
VXBAJLGYBMTJCY
|
8.4 | IC50 | 34 | Yes | |
TVRXNAHDMVOXOV
|
8.4 | IC50 | 2 | — | |
KLJSQTWPBGAZHQ
|
8.4 | IC50 | 4 | — | |
DDPAPPCCQQJSAP
|
8.4 | IC50 | 9 | — | |
GFPPBUZAOLMYKX
|
8.4 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
8.4 | IC50 | 82 | — | |
NRKPJTBUHZKLGS
|
8.4 | Ki | 9 | — | |
YPJSFIQDRPQLPZ
|
8.4 | Ki | 9 | — | |
ZKCWYMOGNNWACW
|
8.4 | Ki | 4 | — | |
SZQYBGGKUBNKSZ
|
8.3 | IC50 | 5 | — | |
QYLYUTQSYHCBOD
|
8.3 | IC50 | 13 | — | |
CJJMNECGBUPMAV
|
8.3 | IC50 | 8 | Yes | |
HUXYBQXJVXOMKX
|
8.3 | IC50 | 28 | — | |
FKAZCQZUYQPWFL
|
8.3 | IC50 | 2 | — | |
PUZNGRPTWFBCMK
|
8.2 | IC50 | 4 | — | |
CELCCCWTAADGDV
|
8.2 | IC50 | 15 | — | |
CSRROEXIZXVOPU
|
8.2 | IC50 | 4 | — | |
GIMRHZPQMMMJKH
|
8.2 | IC50 | 5 | — | |
IUJJKGUBKGMJDU
|
8.2 | IC50 | 2 | — | |
KOLSEKSFVMGHDV
|
8.2 | IC50 | 12 | — | |
WESLFWSZUGLONY
|
8.2 | IC50 | 4 | — | |
YLWSVZLNZZVTSM
|
8.2 | IC50 | 15 | — | |
ZKDXRFMOHZVXSG
|
8.2 | IC50 | 13 | Yes | |
PNYMCFQCHXFMCI
|
8.2 | IC50 | 2 | — | |
UZQXPHDZFUAMQS
|
8.2 | IC50 | 9 | — | |
ZOJWMCDSTRTTOW
|
8.2 | IC50 | 2 | — | |
GCYXEGSPUDSZJY
|
8.2 | IC50 | 17 | Yes | |
TYSWNLQZLBRNSE
|
8.2 | IC50 | 15 | — | |
VUIXUTVIIOVVHV
|
8.2 | IC50 | 3 | — | |
ZSNHIQTXGFQNBW
|
8.2 | IC50 | 3 | — | |
UPQKBKLECVIXJR
|
8.1 | IC50 | 12 | — | |
OEPMKSHSBUZDIB
|
8.1 | IC50 | 2 | — | |
BNVJXUKXMSVXHJ
|
8.1 | IC50 | 2 | — | |
CGKJOISVQXEPSG
|
8.1 | Ki | 9 | — | |
CQWBHMMWZICZRH
|
8.1 | IC50 | 10 | — | |
JWZMXYSZZSYDGV
|
8.1 | IC50 | 4 | — | |
PUVVKKBHOWNLRX
|
8.1 | IC50 | 2 | — | |
RVKNONNXSNALJV
|
8.1 | IC50 | 21 | — | |
DIASEXMEBNQQHZ
|
8.0 | IC50 | 13 | — | |
FFVIVTCGXATTRT
|
8.0 | IC50 | 4 | — | |
IYNDTACKOAXKBJ
|
8.0 | IC50 | 17 | — | |
OHPFNMNHNRGIBV
|
8.0 | IC50 | 2 | — |