Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QWJMFUIHTVAUCH
|
7.3 | IC50 | 3 | — | |
UCBSOBAEFNVYID
|
7.3 | IC50 | 2 | — | |
WPRFMKAORZZEIZ
|
7.3 | IC50 | 3 | — | |
XBQGLWPUGBREQS
|
7.3 | IC50 | 4 | — | |
YTYPEASDFWXHLK
|
7.3 | IC50 | 3 | — | |
AAAQFGUYHFJNHI
|
7.3 | Kd | 252 | — | |
FLASGTNYMYVYKJ
|
7.3 | IC50 | 3 | — | |
LWGUCDPMTIPABX
|
7.3 | IC50 | 4 | — | |
NBBLMCRKPAWOPH
|
7.3 | IC50 | 3 | — | |
WQRKDXUDKMFKPL
|
7.3 | IC50 | 4 | — | |
ZBZCQXDDHPHITA
|
7.3 | IC50 | 4 | — | |
DDIGBXFXYQBMSG
|
7.3 | IC50 | 3 | — | |
FLLDFQACNKMSRM
|
7.3 | IC50 | 3 | — | |
MVAYDDZVYGANLI
|
7.3 | IC50 | 3 | — | |
OENGVXVRDHPNME
|
7.3 | IC50 | 3 | — | |
PQYXGDZAWKQEEM
|
7.3 | IC50 | 3 | — | |
AREGGTVPTLNTCU
|
7.2 | IC50 | 3 | — | |
HSMCUAMXZNQLSQ
|
7.2 | IC50 | 3 | — | |
OJGGGCDIKGWBSR
|
7.2 | IC50 | 2 | — | |
VUVUVNZRUGEAHB
|
7.2 | IC50 | 5 | — | |
WPRFMKAORZZEIZ
|
7.2 | IC50 | 2 | — | |
YDIQBHXHQQZJQQ
|
7.2 | IC50 | 3 | — | |
YNMSRPUOAQPYLV
|
7.2 | IC50 | 3 | — | |
CQPGVZBZRUVJJZ
|
7.2 | IC50 | 3 | — | |
IFFAPYISKKZOPO
|
7.2 | IC50 | 4 | — | |
OYMMHSBUFOLNEY
|
7.2 | IC50 | 3 | — | |
ZNGYYGUCWRDEAS
|
7.2 | IC50 | 3 | — | |
AWVPNUWHMBPXOU
|
7.2 | Kd | 8 | — | |
OZPNRBXVIUPSDJ
|
7.2 | Kd | 4 | — | |
XDAXVUPUYYWFHA
|
7.2 | IC50 | 3 | — | |
ASFZUTSSNARCOL
|
7.2 | IC50 | 3 | — | |
DNVXATUJJDPFDM
|
7.2 | IC50 | 17 | — | |
OGJPTYDTRCDEJC
|
7.2 | IC50 | 3 | — | |
SJSCJYHUBPKPNG
|
7.2 | IC50 | 3 | — | |
SUIIIOQGACLJMI
|
7.2 | IC50 | 3 | — | |
WCNXRFKEDHKCLC
|
7.2 | IC50 | 3 | — | |
YLEHNGYWUWDXNV
|
7.2 | IC50 | 3 | — | |
ZKVURPUQVABYSC
|
7.2 | IC50 | 3 | — | |
XQGQHZQHQKHLDK
|
7.2 | IC50 | 3 | — | |
BKQJIPRADVVRKL
|
7.2 | IC50 | 3 | — | |
FLLDFQACNKMSRM
|
7.2 | IC50 | 3 | — | |
FTYXFBKWRBABJZ
|
7.2 | IC50 | 3 | — | |
HKECFOZBEGKIAX
|
7.2 | IC50 | 3 | — | |
OYDMPDMTZYTSSQ
|
7.2 | IC50 | 3 | — | |
STHZORHCRFBRIV
|
7.2 | IC50 | 3 | — | |
WSQOJBUQSYKMGG
|
7.2 | IC50 | 2 | — | |
CMEIUJXPMXIULZ
|
7.2 | IC50 | 3 | — | |
FAMCYVZRWHZORW
|
7.2 | IC50 | 3 | — | |
GQXFGAMRIGUNFT
|
7.2 | IC50 | 4 | — | |
JFLRJPGRSNHGAL
|
7.2 | IC50 | 3 | — |