Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WTDQWZPPVBDRKD
|
7.4 | IC50 | 3 | — | |
XOUGFEOTWVNPHI
|
7.4 | IC50 | 3 | — | |
AXKZAOMIZYICQV
|
7.4 | IC50 | 2 | — | |
FTHLNVOKHACXIU
|
7.4 | IC50 | 3 | — | |
QGIHDISRDFTWAD
|
7.4 | IC50 | 3 | — | |
AEOQRVQQPVQSRQ
|
7.4 | IC50 | 3 | — | |
HXGQYSSCVKIEIA
|
7.4 | IC50 | 3 | — | |
KOWPYSXWLGSRKS
|
7.4 | IC50 | 3 | — | |
MVAYDDZVYGANLI
|
7.4 | IC50 | 3 | — | |
PBZMPCXVZAPRES
|
7.4 | IC50 | 3 | — | |
RJPKAAVNTLYQAC
|
7.4 | IC50 | 3 | — | |
SDJOVLUEILKTJF
|
7.4 | Ki | 3 | — | |
FRJGKZLDWJMCPQ
|
7.3 | IC50 | 3 | — | |
IXNBIPCXYOBMSS
|
7.3 | IC50 | 3 | — | |
MDRXOFSNECSECW
|
7.3 | Ki | 3 | — | |
NEUUJGUKAZAFHZ
|
7.3 | IC50 | 3 | — | |
SNXGAWWAXJMADO
|
7.3 | IC50 | 3 | — | |
FEBAVJBCNBJJOC
|
7.3 | IC50 | 2 | — | |
KBQLHGZSZFKGCG
|
7.3 | IC50 | 3 | — | |
OFWSNGJQSBQEOU
|
7.3 | IC50 | 2 | — | |
TUWDLUFFAHHNEF
|
7.3 | IC50 | 3 | — | |
ZQFOFTHJENGQKG
|
7.3 | IC50 | 3 | — | |
JKTAXQJDSRMHSS
|
7.3 | IC50 | 3 | — | |
SJACAKNFJFXOJF
|
7.3 | IC50 | 3 | — | |
SMYPWBHABVYAJK
|
7.3 | IC50 | 3 | — | |
UQMYMWRETIHSGQ
|
7.3 | IC50 | 3 | — | |
XRQOPEVIGOZEJD
|
7.3 | IC50 | 3 | — | |
DNVXATUJJDPFDM
|
7.3 | IC50 | 4 | — | |
MZKIOOQWOZDDMX
|
7.3 | IC50 | 3 | — | |
UZPOOTYPBOTHKT
|
7.3 | IC50 | 3 | — | |
WEWCBQWPGVKVPY
|
7.3 | IC50 | 2 | — | |
SJACAKNFJFXOJF
|
7.3 | IC50 | 2 | — | |
ARWMKZDWGIOCEU
|
7.3 | Kd | 4 | — | |
JVTTVFOTQZIFEV
|
7.3 | IC50 | 3 | — | |
UZPOOTYPBOTHKT
|
7.3 | IC50 | 3 | — | |
WAXXYIQBXWBHKY
|
7.3 | IC50 | 2 | — | |
WQEGQSRMXSLEON
|
7.3 | IC50 | 3 | — | |
NBBLMCRKPAWOPH
|
7.3 | IC50 | 3 | — | |
SLTHVRXQOKFPLI
|
7.3 | IC50 | 3 | — | |
BALJMSOPRQWRAP
|
7.3 | IC50 | 3 | — | |
BHZGECKOYMLRSO
|
7.3 | IC50 | 3 | — | |
DAXLHHYYMDQRCH
|
7.3 | IC50 | 3 | — | |
GQXFGAMRIGUNFT
|
7.3 | IC50 | 4 | — | |
GVCFSBGCJBRHFS
|
7.3 | IC50 | 4 | — | |
HMXDNEFPCAGWPH
|
7.3 | IC50 | 3 | — | |
IEEQBCSZMPIUGM
|
7.3 | IC50 | 3 | — | |
JFPHLFWFVVJKQO
|
7.3 | IC50 | 4 | — | |
MBXHXEWZLTYTML
|
7.3 | IC50 | 3 | — | |
MJTVRIBROYBHIV
|
7.3 | IC50 | 3 | — | |
OQBRSKHYDQIBJE
|
7.3 | IC50 | 3 | — |