Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JTXHXYXYGGEYBL
|
7.5 | Kd | 3 | — | |
RWRYTMPXTGYISG
|
7.5 | IC50 | 3 | — | |
VVPPHMRXPGDFBQ
|
7.5 | IC50 | 3 | — | |
FNDFWBANYDEWBA
|
7.4 | Kd | 3 | — | |
IVJMCRKXIOARPS
|
7.4 | IC50 | 3 | — | |
JADOFDPLHYUWBU
|
7.4 | IC50 | 3 | — | |
KGAKOIGDOIZZOQ
|
7.4 | IC50 | 2 | — | |
KOWPYSXWLGSRKS
|
7.4 | IC50 | 2 | — | |
KOYGJJMRJVPCNS
|
7.4 | IC50 | 3 | — | |
ORTRBMKXQWFMTN
|
7.4 | IC50 | 3 | — | |
QIJUHAIEZZEKSX
|
7.4 | IC50 | 3 | — | |
FMJBUHAFPYWEKA
|
7.4 | IC50 | 3 | — | |
HDHIHYNEQCFQNL
|
7.4 | IC50 | 3 | — | |
HSMCUAMXZNQLSQ
|
7.4 | IC50 | 3 | — | |
NCEJUIVQBWZGMA
|
7.4 | IC50 | 3 | — | |
NJQDQDHZAAGIQX
|
7.4 | IC50 | 3 | — | |
PXTNXIAHIKBHPF
|
7.4 | IC50 | 3 | — | |
RKSYSKOBHCWHKB
|
7.4 | IC50 | 3 | — | |
XYESNEVBCXKVML
|
7.4 | IC50 | 2 | — | |
AIPWZDCZUJGLIF
|
7.4 | IC50 | 3 | — | |
FFMRDJNJHCWRIX
|
7.4 | IC50 | 3 | — | |
VUWJZAUOMZSUEU
|
7.4 | IC50 | 3 | — | |
WODOTYIRVRGFSJ
|
7.4 | IC50 | 3 | — | |
XNRZMTWJFLFRMR
|
7.4 | IC50 | 4 | — | |
ZDYWXTGNQATUAC
|
7.4 | IC50 | 2 | — | |
BTGFLXGQPNRXDH
|
7.4 | IC50 | 3 | — | |
CBNDXTMVECMPGV
|
7.4 | IC50 | 4 | — | |
GAVLMQAIIHDXBG
|
7.4 | IC50 | 2 | — | |
GKMMNQCWGZRQTN
|
7.4 | IC50 | 4 | — | |
GPVRSQMGHNALCJ
|
7.4 | IC50 | 3 | — | |
HQEUJXGKBKBFIW
|
7.4 | IC50 | 3 | — | |
IPDBNDHFDHKHDZ
|
7.4 | IC50 | 3 | — | |
JHVSPUDTTXELLE
|
7.4 | IC50 | 3 | — | |
QLRYSHYUZMZZPY
|
7.4 | IC50 | 3 | — | |
SJSCJYHUBPKPNG
|
7.4 | IC50 | 3 | — | |
ZUEZEQZVGBUYFN
|
7.4 | IC50 | 3 | — | |
PXLJQXYHONWMKB
|
7.4 | IC50 | 3 | — | |
UFFMFBORABJCTA
|
7.4 | Ki | 3 | — | |
WUFYDWKEOKQEEP
|
7.4 | IC50 | 3 | — | |
WYUJMOVTXOPUEX
|
7.4 | IC50 | 4 | — | |
ZORLJXWXFABTPZ
|
7.4 | IC50 | 9 | — | |
SNDFCVARRAHINB
|
7.4 | IC50 | 3 | — | |
ZOVYOHAZPIKVOR
|
7.4 | IC50 | 4 | — | |
AURWSPRKUDZZIW
|
7.4 | IC50 | 3 | — | |
IMXDUOIANVGJIA
|
7.4 | IC50 | 4 | — | |
LMCSAEHKLPKZOO
|
7.4 | IC50 | 3 | — | |
LMYKZDUQLVXDIX
|
7.4 | IC50 | 3 | — | |
NVRXYLMWFKVLJI
|
7.4 | IC50 | 3 | — | |
PYJQEIWIODYCRH
|
7.4 | IC50 | 3 | — | |
RKZATRLAMOOMLN
|
7.4 | IC50 | 2 | — |