Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BQDONWPMBNKZCG
|
7.5 | IC50 | 4 | — | |
GZEDEKFDZMUCGJ
|
7.5 | IC50 | 4 | — | |
ZFJHDWKVFUWKQS
|
7.5 | IC50 | 3 | — | |
CLMSQBWNXNAWOK
|
7.5 | IC50 | 2 | — | |
FLEGAAQBQHISDY
|
7.5 | IC50 | 3 | — | |
GKJNYZBASPYBEP
|
7.5 | IC50 | 3 | — | |
SCYBDERMEWGYSR
|
7.5 | IC50 | 2 | — | |
UVCPBOQPPSLUPY
|
7.5 | IC50 | 3 | — | |
BSZDTJJAUVZTBS
|
7.5 | IC50 | 3 | — | |
BWMCWOZPWHUTGN
|
7.5 | IC50 | 3 | — | |
KVTLTFKBEFZOGC
|
7.5 | IC50 | 3 | — | |
PXLJQXYHONWMKB
|
7.5 | IC50 | 3 | — | |
VVSCZWKYDATSNC
|
7.5 | IC50 | 3 | — | |
XZYFNQNYLMTZIS
|
7.5 | IC50 | 3 | — | |
BHEROPFARKLXOP
|
7.5 | IC50 | 4 | — | |
BRAMSTZRKUJRKS
|
7.5 | IC50 | 4 | — | |
FQEWVABJRCOJBI
|
7.5 | IC50 | 4 | — | |
JNYUGWPUYNNZOZ
|
7.5 | Kd | 3 | — | |
KQIUBFKRUFVQEI
|
7.5 | IC50 | 3 | — | |
LORVKFYVSXATKW
|
7.5 | IC50 | 5 | — | |
LZYVFLZEQAANSW
|
7.5 | IC50 | 3 | — | |
MMMRGZLSUKMQOD
|
7.5 | IC50 | 4 | — | |
PHSQIKIQGFDDEU
|
7.5 | IC50 | 2 | — | |
PPCFYGSMPQKDDM
|
7.5 | IC50 | 3 | — | |
UCOMAESNVXJEIJ
|
7.5 | IC50 | 2 | — | |
WIFZFGUMQICZOO
|
7.5 | IC50 | 3 | — | |
BRAMSTZRKUJRKS
|
7.5 | IC50 | 3 | — | |
BUFWGONUWXTMGP
|
7.5 | IC50 | 3 | — | |
GKJNYZBASPYBEP
|
7.5 | IC50 | 3 | — | |
HNJGEQPWIDZIRC
|
7.5 | IC50 | 3 | — | |
KLKMODXQLGKDKQ
|
7.5 | Ki | 3 | — | |
VLVRBRZAFGCGJV
|
7.5 | IC50 | 3 | — | |
WKDIHLGAKPCUJV
|
7.5 | IC50 | 3 | — | |
CRXLFEZLSZPQMT
|
7.5 | IC50 | 2 | — | |
FRDVUWTYVBTBSE
|
7.5 | IC50 | 3 | — | |
IMBCMESWDHPIDA
|
7.5 | IC50 | 3 | — | |
IOHXSSTYGFWMFM
|
7.5 | IC50 | 3 | — | |
IUUGMLRGSKSQJD
|
7.5 | IC50 | 3 | — | |
NUBBUOMZQPTGKS
|
7.5 | IC50 | 2 | — | |
OIAZLVBSFCYPRC
|
7.5 | IC50 | 2 | — | |
QWMJOPLEXJAKPN
|
7.5 | IC50 | 3 | — | |
QXTHZAMLLIIJHM
|
7.5 | IC50 | 3 | — | |
SCYDFQIUWZYQDE
|
7.5 | IC50 | 3 | — | |
UCJMBWXOKLINTN
|
7.5 | IC50 | 4 | — | |
WEHPZXXDBNJUIG
|
7.5 | IC50 | 3 | — | |
WODOTYIRVRGFSJ
|
7.5 | IC50 | 3 | — | |
FRDRCUWLVRNFIJ
|
7.5 | IC50 | 3 | — | |
GZFJPALDEYOFHA
|
7.5 | Ki | 6 | — | |
HIZNONHBBUUYFX
|
7.5 | IC50 | 4 | — | |
IFLPDVNBLNGRJS
|
7.5 | IC50 | 3 | — |