Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SNIKOFNWYKITGY
|
7.6 | IC50 | 3 | — | |
SSELZXGQLGXCDT
|
7.6 | IC50 | 3 | — | |
VFDAORCFAAAXRV
|
7.6 | IC50 | 3 | — | |
OFFYQYIVOWBZLD
|
7.6 | IC50 | 3 | — | |
BYCJBYOKDKPJQP
|
7.6 | IC50 | 3 | — | |
HKECFOZBEGKIAX
|
7.6 | IC50 | 3 | — | |
KKQGFFSHWVTNMA
|
7.6 | IC50 | 3 | — | |
LEMUMFMXNFTRTL
|
7.6 | IC50 | 3 | — | |
MGLUYQBSWDKFIR
|
7.6 | IC50 | 3 | — | |
MLMDKPAWBXFXNA
|
7.6 | IC50 | 3 | — | |
YSAPPGXSSQEHTA
|
7.6 | IC50 | 3 | — | |
YXHZTVCEXBXXJR
|
7.6 | IC50 | 3 | — | |
ABSZIZKRSYKAPX
|
7.6 | IC50 | 4 | — | |
AMRTUWDHDGIYSC
|
7.6 | IC50 | 3 | — | |
BUFWGONUWXTMGP
|
7.6 | IC50 | 3 | — | |
DVICYEUYFBDIJO
|
7.6 | IC50 | 3 | — | |
JBKUGHMRISDLDL
|
7.6 | IC50 | 3 | — | |
NCLGWTFZOQZNIS
|
7.6 | IC50 | 3 | — | |
QCXJZVDATPNNCE
|
7.6 | IC50 | 3 | — | |
QSLHPKXGYOTUHN
|
7.6 | IC50 | 3 | — | |
QTVSDAUHDJBCAA
|
7.6 | IC50 | 4 | — | |
SXBROIQUJXJPJP
|
7.6 | IC50 | 3 | — | |
WCNXRFKEDHKCLC
|
7.6 | IC50 | 3 | — | |
KDRSWORUPZEOGX
|
7.6 | IC50 | 3 | — | |
SFZBPQNERSUWOW
|
7.6 | IC50 | 3 | — | |
UCTNVNGRNJPSOM
|
7.6 | IC50 | 3 | — | |
XQODQNSFZKRZIC
|
7.6 | Kd | 4 | — | |
CURNKPOFSHNCQW
|
7.6 | IC50 | 2 | — | |
DHQSSAHSRGVRJY
|
7.6 | IC50 | 3 | — | |
FFHFKSXIZXKTRE
|
7.6 | IC50 | 3 | — | |
FUOUPXXFTDVPGM
|
7.6 | IC50 | 3 | — | |
GTFJSDPFUPQADT
|
7.6 | IC50 | 2 | — | |
NMPGZGXWNHOBFF
|
7.6 | IC50 | 3 | — | |
UCTNVNGRNJPSOM
|
7.6 | IC50 | 3 | — | |
CPWCZLPJMXCWDY
|
7.6 | IC50 | 3 | — | |
FZFLGRAVZYFGBB
|
7.6 | Kd | 4 | — | |
FDMPGPNYXCYCQJ
|
7.5 | IC50 | 3 | — | |
KQIUBFKRUFVQEI
|
7.5 | IC50 | 3 | — | |
QLRYSHYUZMZZPY
|
7.5 | IC50 | 4 | — | |
RLAHXCWDADVADO
|
7.5 | IC50 | 4 | — | |
TUWDLUFFAHHNEF
|
7.5 | IC50 | 3 | — | |
VFDAORCFAAAXRV
|
7.5 | IC50 | 3 | — | |
WQBRHFBWJUCVRR
|
7.5 | IC50 | 3 | — | |
FESHYOISGIZOBW
|
7.5 | IC50 | 2 | — | |
IYRDZCVNOKVDNI
|
7.5 | IC50 | 3 | — | |
SUFVOUWYHJXPBW
|
7.5 | Kd | 4 | — | |
UAEXWMVCHTWKPO
|
7.5 | IC50 | 2 | — | |
UHWGSUFICDUCKV
|
7.5 | IC50 | 3 | — | |
VVRZMYLMDPVHTL
|
7.5 | Ki | 3 | — | |
ZSBDKRBBDNFMHY
|
7.5 | Ki | 3 | — |