Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FKTRRXZUNCKQOU
|
7.7 | IC50 | 3 | — | |
OJCRNHCUTYXXFI
|
7.7 | Kd | 3 | — | |
PXGREUPWZAUELV
|
7.7 | IC50 | 3 | — | |
RIDHDDTVNQHKEQ
|
7.7 | IC50 | 3 | — | |
SSELZXGQLGXCDT
|
7.7 | IC50 | 2 | — | |
YAJRUKJDKBVQBZ
|
7.7 | IC50 | 3 | — | |
YJEIXSZAEKFWTM
|
7.7 | IC50 | 3 | — | |
RYGFKPUPLGKCHY
|
7.7 | IC50 | 3 | — | |
CHBGVONAUISDSX
|
7.7 | IC50 | 3 | — | |
FLEGAAQBQHISDY
|
7.7 | IC50 | 3 | — | |
GLMGIYSAZNFOHX
|
7.7 | IC50 | 3 | — | |
JKLFTZFZNNCDAE
|
7.7 | IC50 | 4 | — | |
KDVBPVJMVKBRPB
|
7.7 | IC50 | 2 | — | |
OGJPTYDTRCDEJC
|
7.7 | IC50 | 3 | — | |
SAJVWIFFPNLZRK
|
7.7 | IC50 | 2 | — | |
USNVRJYSAUJTNT
|
7.7 | IC50 | 4 | — | |
XMRBIQDRTZCVGG
|
7.7 | IC50 | 3 | — | |
IZWQPEYVFYWESQ
|
7.7 | IC50 | 3 | — | |
CSMGGKQPASRAIQ
|
7.7 | IC50 | 3 | — | |
GAFAVXVVQUWUQX
|
7.7 | IC50 | 3 | — | |
GLMGIYSAZNFOHX
|
7.7 | IC50 | 3 | — | |
HMRUYZVXBSSKBX
|
7.7 | IC50 | 3 | — | |
IAYAEBUJIVBSPF
|
7.7 | IC50 | 2 | — | |
KILRLNJOBPEYAV
|
7.7 | IC50 | 3 | — | |
KKLVVGZXBWABFO
|
7.7 | IC50 | 3 | — | |
LLRPIXCDTAUFLE
|
7.7 | IC50 | 4 | — | |
MRXGSXIGPZYETN
|
7.7 | IC50 | 3 | — | |
POKZINYHLOHGEB
|
7.7 | Kd | 4 | — | |
TWYGARCNNFAUNW
|
7.7 | IC50 | 3 | — | |
UQMYMWRETIHSGQ
|
7.7 | IC50 | 3 | — | |
UYRUHHLEYUGTMC
|
7.7 | IC50 | 3 | — | |
ZDMWQHIIHYYGIB
|
7.7 | IC50 | 3 | — | |
KLPMURBFDSDZSU
|
7.7 | IC50 | 3 | — | |
GTLGKZJPNAWIBT
|
7.7 | IC50 | 3 | — | |
JSKLBERKQHGHCP
|
7.7 | IC50 | 3 | — | |
LMQMHIFIMOPETK
|
7.7 | IC50 | 3 | — | |
NAPOLFVZKFHOBG
|
7.7 | IC50 | 4 | — | |
OCOWZEOSBFUWRU
|
7.7 | IC50 | 2 | — | |
WQEGQSRMXSLEON
|
7.7 | IC50 | 4 | — | |
XZYFNQNYLMTZIS
|
7.7 | IC50 | 3 | — | |
IFLPDVNBLNGRJS
|
7.7 | IC50 | 3 | — | |
HQEUJXGKBKBFIW
|
7.6 | IC50 | 3 | — | |
JQGLKQWMMRCIIG
|
7.6 | IC50 | 4 | — | |
LDQWWSKUZGJSPQ
|
7.6 | IC50 | 2 | — | |
MYTABVRHXGACGI
|
7.6 | IC50 | 4 | — | |
OMLHQPIYXLWGGG
|
7.6 | IC50 | 3 | — | |
OZSRLNZYSOUOCT
|
7.6 | IC50 | 3 | — | |
PKHUSSXCMLLVRI
|
7.6 | IC50 | 3 | — | |
PKWSPAGTIXNWLL
|
7.6 | IC50 | 3 | — | |
QDMDJWBTMQQUPC
|
7.6 | IC50 | 3 | — |