Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IBRUPFNOCSUECL
|
7.8 | IC50 | 3 | — | |
KJMPMBQYOMBJLE
|
7.8 | IC50 | 3 | — | |
OGVXCCMPKKUNFP
|
7.8 | IC50 | 3 | — | |
RDWRDUFEWMSPGQ
|
7.8 | Kd | 4 | — | |
VBNIZIAZOQSIGW
|
7.8 | IC50 | 2 | — | |
XMRBIQDRTZCVGG
|
7.8 | IC50 | 3 | — | |
YORKSQKTPMJQBD
|
7.8 | IC50 | 3 | — | |
ZBKQIKDKLUJFMK
|
7.8 | Ki | 3 | — | |
ZJTYXGWJNWESQV
|
7.8 | Kd | 3 | — | |
AVWFNEVSOVPOLY
|
7.8 | IC50 | 3 | — | |
AVWFNEVSOVPOLY
|
7.8 | IC50 | 3 | — | |
FZOWBAIZBAZQAF
|
7.8 | IC50 | 2 | — | |
KVPRUGZKNCVUEL
|
7.8 | IC50 | 2 | — | |
LZQJKADDYCLNSB
|
7.8 | IC50 | 2 | — | |
MGLUYQBSWDKFIR
|
7.8 | IC50 | 3 | — | |
NRKGWEXMFVBBBE
|
7.8 | IC50 | 3 | — | |
WVDZBUCUXBEFHG
|
7.8 | IC50 | 3 | — | |
YJEIXSZAEKFWTM
|
7.8 | IC50 | 3 | — | |
BYVIHYLKGUPNHK
|
7.8 | IC50 | 3 | — | |
GTYWOEFUZYKPQR
|
7.8 | IC50 | 3 | — | |
JMENTVKUBOUMCJ
|
7.8 | IC50 | 3 | — | |
LOOFPBVYOVHBCL
|
7.8 | IC50 | 3 | — | |
NDEORODKVUYMFQ
|
7.8 | Kd | 9 | — | |
PDCBJZVPIGAEBL
|
7.8 | IC50 | 4 | — | |
QXUMXOZTPSIGSM
|
7.8 | IC50 | 3 | — | |
RCXOWIAUDIGVEW
|
7.8 | IC50 | 2 | — | |
RGKUFEQXYKVMOO
|
7.8 | IC50 | 4 | — | |
RPBWYZZANXCAJX
|
7.8 | IC50 | 3 | — | |
SCOGYYPZUPWMLU
|
7.8 | IC50 | 3 | — | |
SNQJYZHFKZPJDR
|
7.8 | IC50 | 2 | — | |
SVEGTFMYOXJKMY
|
7.8 | IC50 | 3 | — | |
ZLVIFBCNFIAMBN
|
7.8 | IC50 | 3 | — | |
CBNDXTMVECMPGV
|
7.8 | IC50 | 4 | — | |
DGXUFGAFFVEFEU
|
7.8 | IC50 | 3 | — | |
DVNSWDWISPDNHZ
|
7.8 | IC50 | 3 | — | |
FOEVWVKNXOCNTG
|
7.8 | IC50 | 3 | — | |
NGGZYQVCSSIVJR
|
7.8 | IC50 | 2 | — | |
NHQWTZLQTWSZGU
|
7.8 | IC50 | 4 | — | |
NMPGZGXWNHOBFF
|
7.8 | IC50 | 3 | — | |
OSOMHZBGIZCTKM
|
7.8 | IC50 | 4 | — | |
RJDVRXGILIWOCC
|
7.8 | IC50 | 2 | — | |
YSAPPGXSSQEHTA
|
7.8 | IC50 | 3 | — | |
RGHQRULWHKEQHE
|
7.8 | IC50 | 3 | — | |
AYMBFUSITNSKHY
|
7.7 | IC50 | 3 | — | |
DVNSWDWISPDNHZ
|
7.7 | IC50 | 3 | — | |
MVALXNVRFKZEQJ
|
7.7 | IC50 | 2 | — | |
SWZWWWDWBVBZDV
|
7.7 | IC50 | 3 | — | |
WGJDGQSSFHDLIX
|
7.7 | IC50 | 3 | — | |
XSISVIBLCIAEGR
|
7.7 | IC50 | 4 | — | |
CYZNNGBIFDNKBV
|
7.7 | IC50 | 2 | — |