Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DLEHIPJVRSZXAI
|
8.1 | Ki | 3 | — | |
WSHVXKCBHNIVJO
|
8.1 | IC50 | 4 | — | |
HSYFXAZMBHUTJZ
|
8.0 | Ki | 3 | — | |
LJLJARSDBHJRGG
|
8.0 | Ki | 4 | — | |
UNODBAFOZVBZBF
|
8.0 | Ki | 4 | — | |
UXFXOEGGFKVCDW
|
8.0 | IC50 | 4 | — | |
ZJXAVKZXYZJJKO
|
8.0 | IC50 | 3 | — | |
WHDUHJYPRJXLGF
|
8.0 | Kd | 4 | — | |
GNMUEVRJHCWKTO
|
8.0 | Ki | 3 | — | |
JBPWXWQIGDWQHR
|
8.0 | IC50 | 15 | — | |
KJSPRHSFQGRYOT
|
8.0 | IC50 | 3 | — | |
RIDHDDTVNQHKEQ
|
8.0 | IC50 | 3 | — | |
ZZJIAOWVSKZQGQ
|
8.0 | IC50 | 3 | — | |
QSRRNUBIKNVQHO
|
7.9 | IC50 | 4 | — | |
BSZDTJJAUVZTBS
|
7.9 | IC50 | 2 | — | |
FBYKSRDDFYPNNO
|
7.9 | IC50 | 3 | — | |
GQVNARRVGGOXNP
|
7.9 | IC50 | 2 | — | |
GQVNARRVGGOXNP
|
7.9 | IC50 | 3 | — | |
KVTLTFKBEFZOGC
|
7.9 | IC50 | 2 | — | |
NBJPFMDWXKYTQF
|
7.9 | IC50 | 2 | — | |
NCLGWTFZOQZNIS
|
7.9 | IC50 | 3 | — | |
NPLFXOGRUJPLAA
|
7.9 | IC50 | 3 | — | |
PBUQLYYLOVDBLR
|
7.9 | IC50 | 3 | — | |
RCXOWIAUDIGVEW
|
7.9 | IC50 | 2 | — | |
RDONXGFGWSSFMY
|
7.9 | Ki | 6 | — | |
WGJDGQSSFHDLIX
|
7.9 | IC50 | 2 | — | |
YORKSQKTPMJQBD
|
7.9 | IC50 | 2 | — | |
ZBIYSSHSZQVNSP
|
7.9 | IC50 | 2 | — | |
KNBYFXZNSOENGW
|
7.9 | Kd | 5 | — | |
ZYJNOYAZLFPWBD
|
7.9 | IC50 | 4 | — | |
CRYAUTCZOKUESS
|
7.9 | IC50 | 2 | — | |
FBYKSRDDFYPNNO
|
7.9 | IC50 | 3 | — | |
IPYPJQJYDYFZCL
|
7.9 | IC50 | 3 | — | |
IYRDZCVNOKVDNI
|
7.9 | IC50 | 2 | — | |
JBWFCYLPISSKIG
|
7.9 | IC50 | 3 | — | |
JRPLDEULPIHXGO
|
7.9 | IC50 | 3 | — | |
MVALXNVRFKZEQJ
|
7.9 | IC50 | 2 | — | |
NEOVBISHUWMCQM
|
7.9 | IC50 | 3 | — | |
OQBRSKHYDQIBJE
|
7.9 | IC50 | 2 | — | |
RJVJSMKBCOIXKN
|
7.9 | IC50 | 3 | — | |
SMYPWBHABVYAJK
|
7.9 | IC50 | 2 | — | |
TUXHCXODKHDHKT
|
7.9 | IC50 | 2 | — | |
VLVRBRZAFGCGJV
|
7.9 | IC50 | 3 | — | |
XOEVAYXDSJABMS
|
7.9 | Ki | 3 | — | |
YDFGIFLYGLMJSV
|
7.9 | IC50 | 4 | — | |
ZZJIAOWVSKZQGQ
|
7.9 | IC50 | 3 | — | |
NWYXVTBJGUHMRR
|
7.9 | Kd | 3 | — | |
ASOYBTGQKMWPGU
|
7.8 | IC50 | 3 | — | |
BRBCSVDUUHHTIS
|
7.8 | IC50 | 4 | — | |
DDRRENHDNHGPEG
|
7.8 | IC50 | 3 | — |