Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XYFBFOQWZFRJRE
|
6.2 | IC50 | 3 | — | |
ZQXOBYVSSHZKCM
|
6.2 | IC50 | 2 | — | |
HONVADOKRZTBCS
|
6.2 | IC50 | 2 | — | |
LBELIXDRRWMQKV
|
6.2 | IC50 | 3 | — | |
ONUKWYBZXUKVSG
|
6.2 | IC50 | 3 | — | |
PAXZSBFZQIWSKA
|
6.2 | IC50 | 2 | — | |
COGXANVMWYYUMM
|
6.2 | Ki | 2 | — | |
RUVPNJSJTWTANE
|
6.1 | IC50 | 2 | — | |
SGTFNLMVIRZWTA
|
6.1 | IC50 | 2 | — | |
CIBHWLGHOAYWGR
|
6.1 | IC50 | 2 | — | |
BURYFVYAIGGHQI
|
6.1 | IC50 | 3 | — | |
GWZFTXQVWCWFJG
|
6.1 | IC50 | 3 | — | |
MGCJPZAHHFJYBA
|
6.1 | IC50 | 3 | — | |
OUZWCWPWAOUTBA
|
6.1 | IC50 | 2 | — | |
WHZNMFZHYFFFQG
|
6.1 | IC50 | 2 | — | |
FYEHQUXVXRMVBS
|
6.1 | IC50 | 2 | — | |
NIFODZUHQBXOII
|
6.1 | IC50 | 6 | — | |
FRNOWHXMMCGFDO
|
6.0 | IC50 | 2 | — | |
KKNOUVNOCNNTDD
|
6.0 | IC50 | 2 | — | |
DRXUCZBMTLNYCO
|
6.0 | IC50 | 2 | — | |
HSOYFUMYVDSCGZ
|
6.0 | IC50 | 2 | — | |
KQMNYLGXKJUKRF
|
6.0 | IC50 | 2 | — | |
KXXIBIBXJMYWNL
|
6.0 | Kd | 4 | — | |
LNAXUPYBJSUPHK
|
6.0 | IC50 | 2 | — | |
LOCYBPVGKQMTII
|
6.0 | IC50 | 2 | — | |
ULDFEUPLPPWJDA
|
6.0 | IC50 | 3 | — | |
YIIAEOSGRYXGSO
|
6.0 | IC50 | 2 | — |