Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VYWGWQXJWULHNO
|
6.6 | IC50 | 3 | — | |
WEXADKQIKVPYMF
|
6.6 | IC50 | 3 | — | |
ZJANGOZVQMLDFN
|
6.6 | IC50 | 3 | — | |
SCAMMXNLCDAQKQ
|
6.6 | IC50 | 3 | — | |
ASTXGKOUBPCCPU
|
6.5 | IC50 | 3 | — | |
SBDOCCVDBJLSLR
|
6.5 | IC50 | 3 | — | |
WPHNAFYBBIAYKY
|
6.5 | IC50 | 3 | — | |
XNUKXIGJCJJBQX
|
6.5 | IC50 | 3 | — | |
JGGBFOUTSJEGRT
|
6.5 | Ki | 4 | — | |
UCVZNFYFNWAPFX
|
6.5 | IC50 | 3 | — | |
XLMQZASMJFSBJQ
|
6.5 | IC50 | 3 | — | |
BHUOTMULUBCHII
|
6.5 | IC50 | 3 | — | |
HHLPOWRWLBEWKR
|
6.5 | IC50 | 3 | — | |
KBDDUZVOHAQRGN
|
6.5 | IC50 | 3 | — | |
PXXDOEMDQBOWHE
|
6.5 | IC50 | 3 | — | |
ULNHSRPVGJEURD
|
6.5 | IC50 | 4 | — | |
GFVREQSKPNZXLD
|
6.5 | IC50 | 3 | — | |
QGSWOCCDAUKNAQ
|
6.5 | Ki | 3 | — | |
ZMFIMBNRJYXBHU
|
6.4 | IC50 | 3 | — | |
BYXLVMRVUBFJJF
|
6.4 | IC50 | 3 | — | |
RZLGXMUFJRNCFA
|
6.4 | IC50 | 3 | — | |
VKGQTQLKCFTHGK
|
6.4 | IC50 | 2 | — | |
VOXWVXCIJOFLCE
|
6.4 | IC50 | 4 | — | |
NCPRCNJIGPDNGS
|
6.4 | Ki | 3 | — | |
DPBKLIVPNYGQQG
|
6.4 | Kd | 3 | — | |
RWLWADJBUXMBKV
|
6.4 | IC50 | 3 | — | |
WVDIPPMCQKBWHV
|
6.3 | IC50 | 2 | — | |
VJPKOWZJHFRYJT
|
6.3 | IC50 | 3 | — | |
GVLMPZNONRSUIH
|
6.3 | IC50 | 3 | — | |
NVUCJVXTEMYIJR
|
6.3 | IC50 | 3 | — | |
BZNFHPBYRCLAHN
|
6.3 | IC50 | 2 | — | |
HXJWEYPXEZZATP
|
6.3 | IC50 | 3 | — | |
KPXUTHWBDFMTIF
|
6.3 | IC50 | 3 | — | |
LEGSCEIDRZQSRJ
|
6.3 | IC50 | 3 | — | |
LSWFCIPBUIBLDW
|
6.3 | IC50 | 3 | — | |
LWXZPBREHHJQDV
|
6.3 | IC50 | 3 | — | |
OWUQUQCSBQATFQ
|
6.3 | IC50 | 2 | — | |
UBIAANPPYMMVSI
|
6.3 | IC50 | 2 | — | |
UJPOOIUOVCPCTL
|
6.3 | IC50 | 4 | — | |
VQFWLAVCHMSMML
|
6.3 | IC50 | 3 | — | |
YIIAEOSGRYXGSO
|
6.3 | IC50 | 2 | — | |
YTFPNQZFSVSZGW
|
6.3 | IC50 | 3 | — | |
LPLJCQTWKUNXIE
|
6.3 | IC50 | 3 | — | |
YGKMNXJMNMMORF
|
6.3 | Ki | 3 | — | |
KJLXKCQTAXTWLF
|
6.2 | IC50 | 3 | — | |
SKDNDJWEBPQKCS
|
6.2 | Kd | 5 | — | |
IZLQRTZZHBLSKO
|
6.2 | IC50 | 6 | — | |
WXZFQCVRGXOYGQ
|
6.2 | IC50 | 3 | — | |
OOPLGRXMPNAWKN
|
6.2 | IC50 | 3 | — | |
KRQNRCGKZXQJBI
|
6.2 | IC50 | 2 | — |