Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JCMVYYCXZAYXHK
|
6.8 | IC50 | 3 | — | |
MLQZIRMMNHSJKH
|
6.8 | IC50 | 3 | — | |
PIPFCKKGOLUZIH
|
6.8 | IC50 | 3 | — | |
RFBMWIYVIXUMRE
|
6.8 | IC50 | 3 | — | |
DTIQMIRHDCHPIP
|
6.8 | IC50 | 3 | — | |
BIQYOSNHGNQSTQ
|
6.8 | IC50 | 3 | — | |
CPMTVMSTJKIGJI
|
6.8 | IC50 | 4 | — | |
FAMCYVZRWHZORW
|
6.8 | IC50 | 3 | — | |
KILRLNJOBPEYAV
|
6.8 | IC50 | 3 | — | |
MJNSUGCWCAGANT
|
6.8 | IC50 | 3 | — | |
DDCDPEKGXFRTDS
|
6.8 | IC50 | 3 | — | |
GXKIVKDALCGWBS
|
6.8 | IC50 | 3 | — | |
JVAKWUYUZCOCKR
|
6.8 | IC50 | 4 | — | |
PYQBVMHZKQXFAY
|
6.8 | IC50 | 3 | — | |
QKILPYXMYOTNIL
|
6.8 | IC50 | 3 | — | |
RSMYFSPOTCDHHJ
|
6.8 | Ki | 5 | — | |
SOSVCXWWZFMQQP
|
6.8 | IC50 | 3 | — | |
XKUUHELVHBNAMN
|
6.8 | IC50 | 3 | — | |
YHZBCBREIIKZHU
|
6.8 | IC50 | 3 | — | |
GAORTSKVVPSHRF
|
6.8 | IC50 | 3 | — | |
JEBJXGHLBZQKNY
|
6.8 | IC50 | 3 | — | |
WZPMLZHTAAYDCQ
|
6.8 | IC50 | 3 | — | |
ZSGFXTRWCMGRPZ
|
6.8 | IC50 | 3 | — | |
AGXHDPYHRCHDBA
|
6.7 | IC50 | 3 | — | |
SSCBXXKTZLTDDN
|
6.7 | IC50 | 3 | — | |
WMLLDTCULACFBH
|
6.7 | IC50 | 3 | — | |
BFDSCBNQKZOCJH
|
6.7 | IC50 | 2 | — | |
CLDFWWPJBAFFIK
|
6.7 | IC50 | 3 | — | |
IXWMDWQZYYSEGS
|
6.7 | IC50 | 3 | — | |
AWTFSKPTZUHXSW
|
6.7 | IC50 | 3 | — | |
BRQOWLMNQSLGPU
|
6.7 | IC50 | 3 | — | |
JKUNIMOTGXIVSR
|
6.7 | IC50 | 3 | — | |
JNYUGWPUYNNZOZ
|
6.7 | IC50 | 4 | — | |
MPDWALFCXGTZJW
|
6.7 | IC50 | 3 | — | |
NGXAMXNWIHBLBN
|
6.7 | Kd | 6 | — | |
NTQVJGUGYLGXNI
|
6.7 | IC50 | 3 | — | |
VBWJYWJSBHIBOW
|
6.7 | IC50 | 3 | — | |
VJIUYADBWVTBNH
|
6.7 | IC50 | 3 | — | |
NETXMUIMUZJUTB
|
6.7 | IC50 | 4 | — | |
SGQSLPKSTYGKNO
|
6.7 | IC50 | 3 | — | |
WGVAADOVZXANRM
|
6.7 | IC50 | 3 | — | |
ZUTVFNRARULPEX
|
6.7 | IC50 | 2 | — | |
IJUSAWCETGWNEQ
|
6.7 | IC50 | 3 | — | |
XITXIIWQQYIONX
|
6.7 | IC50 | 3 | — | |
FBLOSBSWOXHYPV
|
6.6 | IC50 | 3 | — | |
PLMVDZBEQUQDAZ
|
6.6 | IC50 | 2 | — | |
JESIANVRZVTARG
|
6.6 | IC50 | 2 | — | |
QUHZSJOJWWZZCP
|
6.6 | IC50 | 4 | — | |
DXUMILREMTTZQK
|
6.6 | IC50 | 3 | — | |
FSMTUHGXWGJNKK
|
6.6 | IC50 | 4 | — |