Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FRBRZGLUFOZRGD
|
7.0 | IC50 | 4 | — | |
JUNKHWUBWMACDY
|
7.0 | IC50 | 3 | — | |
LHEGCVROQQOOOL
|
7.0 | IC50 | 3 | — | |
MTBDHPJCWYLCBM
|
7.0 | IC50 | 7 | — | |
NLJFSVIZSWAERX
|
7.0 | IC50 | 3 | — | |
OVLDCYAZEIXCEQ
|
7.0 | IC50 | 4 | — | |
STSKCRDOTKSTPF
|
7.0 | IC50 | 3 | — | |
WHSDNSXIFWGGOD
|
7.0 | IC50 | 4 | — | |
YINBDXKXEYUKBO
|
7.0 | IC50 | 3 | — | |
JUNKHWUBWMACDY
|
7.0 | IC50 | 3 | — | |
GAFYFVRFEKFZOU
|
7.0 | IC50 | 4 | — | |
HBIBLLVDGBUKCQ
|
7.0 | IC50 | 4 | — | |
IMUJKGKBDBVTGZ
|
7.0 | IC50 | 3 | — | |
MWVVALQFXSOQLF
|
7.0 | IC50 | 3 | — | |
QNOJAPBYTXGBLX
|
7.0 | Ki | 5 | — | |
UXOOYKGHOJVFQB
|
7.0 | IC50 | 3 | — | |
XFGHSUSRHXWNEX
|
7.0 | IC50 | 3 | — | |
OABQDWQBXSGEDG
|
7.0 | IC50 | 9 | — | |
PTAMRJLIOCHJMQ
|
6.9 | Kd | 6 | — | |
RQSRLTLIMDDPDM
|
6.9 | IC50 | 4 | — | |
SVWVGWHDUPYUFQ
|
6.9 | IC50 | 4 | — | |
IHOWNNYVAUSWOU
|
6.9 | IC50 | 7 | — | |
SDIHFORMFMHWNK
|
6.9 | IC50 | 6 | — | |
IKGRWYRGRUJEIF
|
6.9 | IC50 | 3 | — | |
KRBXHYJZXGUPRJ
|
6.9 | IC50 | 3 | — | |
NKRWXLLSKYGFGB
|
6.9 | IC50 | 3 | — | |
OCRZEXONTRGXJJ
|
6.9 | Kd | 3 | — | |
PIPFCKKGOLUZIH
|
6.9 | IC50 | 3 | — | |
PIWFRDGCNFFYEO
|
6.9 | IC50 | 3 | — | |
QXYGIHZVXILREV
|
6.9 | IC50 | 3 | — | |
XCGFXDCZVZODBT
|
6.9 | IC50 | 3 | — | |
YXHZTVCEXBXXJR
|
6.9 | IC50 | 3 | — | |
ZFCPBFSCVUQCLF
|
6.9 | IC50 | 3 | — | |
ZLFZRGHIIRSEBW
|
6.9 | IC50 | 3 | — | |
XOCKWBJNBUYYAL
|
6.9 | IC50 | 5 | — | |
SMYWDSZXWMKRLF
|
6.9 | IC50 | 3 | — | |
AQMPZYCOHRMIPG
|
6.9 | IC50 | 3 | — | |
BDBFPELIWNNUAS
|
6.9 | IC50 | 3 | — | |
CWZBKMRDRUFOGI
|
6.9 | IC50 | 3 | — | |
LKHKHWRBQLPSBP
|
6.9 | IC50 | 3 | — | |
LPQLUGIBIOVXPF
|
6.9 | IC50 | 3 | — | |
MPUJMCAEPNAZNL
|
6.9 | IC50 | 3 | — | |
PEROKLOUIURSIS
|
6.9 | IC50 | 3 | — | |
RJCJQUKBDBNIOB
|
6.9 | IC50 | 4 | — | |
UGVSWFJGRKHVMD
|
6.9 | IC50 | 4 | — | |
WKAWRKNMCTXBMF
|
6.9 | IC50 | 3 | — | |
NVUCJVXTEMYIJR
|
6.9 | IC50 | 3 | — | |
HFXQHVKVUNQRBN
|
6.9 | IC50 | 7 | — | |
GHYCWVRIEDGGFQ
|
6.8 | IC50 | 4 | — | |
HDFQNQPMGAHQTL
|
6.8 | IC50 | 5 | — |