Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NHUYOZGLCLQXEB
|
7.1 | IC50 | 3 | — | |
PASBWKAEFYVJHG
|
7.1 | IC50 | 3 | — | |
VAXZYGLGDOWBGT
|
7.1 | IC50 | 3 | — | |
VLEMFHFORYINCB
|
7.1 | IC50 | 4 | — | |
KXSJLOFFUFDGTE
|
7.1 | IC50 | 6 | — | |
LCXHXIMNUYTCEI
|
7.1 | IC50 | 3 | — | |
HXVTYKVZGFHITR
|
7.1 | IC50 | 3 | — | |
IVXYIGADMWHQDD
|
7.1 | IC50 | 4 | — | |
SRFOIWNXIILSNJ
|
7.1 | IC50 | 4 | — | |
XSOFZNARGSJIQN
|
7.1 | IC50 | 4 | — | |
ZAIFEOJGYZIMNX
|
7.1 | IC50 | 3 | — | |
BVDVIORIEDCJPV
|
7.1 | IC50 | 3 | — | |
DUZXHNLPDHPTHC
|
7.1 | IC50 | 3 | — | |
GFDDTDKCZCGJLM
|
7.1 | Kd | 5 | — | |
IITSESCLMNYTBQ
|
7.1 | IC50 | 3 | — | |
MZKIOOQWOZDDMX
|
7.1 | IC50 | 3 | — | |
QIJUHAIEZZEKSX
|
7.1 | IC50 | 3 | — | |
WVDZBUCUXBEFHG
|
7.1 | IC50 | 3 | — | |
XJIIOIPLGWEZJR
|
7.1 | Ki | 3 | — | |
BWECVGNIEMDNMY
|
7.0 | IC50 | 2 | — | |
GKMMNQCWGZRQTN
|
7.0 | IC50 | 2 | — | |
KUCAMLWGYMEYGQ
|
7.0 | IC50 | 3 | — | |
OBZUUWUBOOUBNE
|
7.0 | IC50 | 7 | — | |
OGSOMZCUMMDDJU
|
7.0 | IC50 | 4 | — | |
PYJQEIWIODYCRH
|
7.0 | IC50 | 3 | — | |
WUFYDWKEOKQEEP
|
7.0 | IC50 | 3 | — | |
YAUNGVSDDBLIPR
|
7.0 | IC50 | 3 | — | |
IKKUVCXGUJTONF
|
7.0 | IC50 | 6 | — | |
LCXHXIMNUYTCEI
|
7.0 | IC50 | 3 | — | |
OXYDGMKIFXNGOS
|
7.0 | IC50 | 3 | — | |
QNRNHBQTJGHZSO
|
7.0 | IC50 | 3 | — | |
AAFNIAPCKWGXDG
|
7.0 | IC50 | 3 | — | |
BKDMSQCDGPSQFW
|
7.0 | IC50 | 3 | — | |
CFUYRGUSQPAALN
|
7.0 | IC50 | 3 | — | |
KOSOJYPHXKHVFL
|
7.0 | IC50 | 3 | — | |
LMLJGVCFCYGAST
|
7.0 | IC50 | 3 | — | |
BHHISRQWOKUVFO
|
7.0 | IC50 | 3 | — | |
HQWHFYOMOHBRTB
|
7.0 | Ki | 3 | — | |
IQIUDSWFPYGIST
|
7.0 | IC50 | 3 | — | |
NYYPYDLZLGCKOU
|
7.0 | IC50 | 4 | — | |
XASDFFVVUGREBP
|
7.0 | IC50 | 3 | — | |
XPDXANVGYAEATN
|
7.0 | IC50 | 3 | — | |
FRBRZGLUFOZRGD
|
7.0 | IC50 | 5 | — | |
FTYXFBKWRBABJZ
|
7.0 | IC50 | 3 | — | |
HXENBKGGEPBXOQ
|
7.0 | IC50 | 3 | — | |
JSJHNZMAOMLIME
|
7.0 | IC50 | 3 | — | |
RTFLOGJKYBGANO
|
7.0 | IC50 | 4 | — | |
AMGMXABLUGQVQD
|
7.0 | IC50 | 3 | — | |
AQMPZYCOHRMIPG
|
7.0 | IC50 | 3 | — | |
BNWMHKNZCUUJMF
|
7.0 | IC50 | 3 | — |