Target Details
| UniProt AC | Q15059 |
|---|---|
| Gene Symbol | BRD3 |
| Protein Name | Bromodomain-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 727
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (727)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SDLMPYCGZKLARA
|
7.2 | IC50 | 4 | — | |
ZQTWZFDWESQAJC
|
7.2 | IC50 | 4 | — | |
FFHFKSXIZXKTRE
|
7.2 | IC50 | 3 | — | |
IMXDUOIANVGJIA
|
7.2 | IC50 | 3 | — | |
LFNLJQQQSRYUHQ
|
7.2 | IC50 | 3 | — | |
SSCBXXKTZLTDDN
|
7.2 | IC50 | 3 | — | |
XNRZMTWJFLFRMR
|
7.2 | IC50 | 3 | — | |
DNVXATUJJDPFDM
|
7.2 | IC50 | 4 | — | |
FUOUPXXFTDVPGM
|
7.2 | IC50 | 3 | — | |
JLNZMTDBARFXJN
|
7.2 | Kd | 9 | — | |
LRWGLQDVNJOJKQ
|
7.2 | IC50 | 3 | — | |
IBJLUHJBIGMOMD
|
7.2 | IC50 | 4 | — | |
LTGAYVZNSVTKFS
|
7.2 | IC50 | 3 | — | |
BNWMHKNZCUUJMF
|
7.1 | IC50 | 3 | — | |
FUXOAMWDPVPAFQ
|
7.1 | IC50 | 3 | — | |
IMYHVLQAXUTNRG
|
7.1 | IC50 | 3 | — | |
QZZCUOVXHPAQRQ
|
7.1 | IC50 | 5 | — | |
SKTNIECRSURWAZ
|
7.1 | IC50 | 3 | — | |
STEDHESXTGJFOX
|
7.1 | IC50 | 3 | — | |
AREGGTVPTLNTCU
|
7.1 | IC50 | 3 | — | |
ITQINGMSTPZGFO
|
7.1 | IC50 | 3 | — | |
PXGREUPWZAUELV
|
7.1 | IC50 | 3 | — | |
PXGREUPWZAUELV
|
7.1 | IC50 | 3 | — | |
FQEWVABJRCOJBI
|
7.1 | IC50 | 3 | — | |
MHDJYXZJVBCMGS
|
7.1 | IC50 | 3 | — | |
MSZSAGAHXQKHRZ
|
7.1 | IC50 | 3 | — | |
MTKZUOYFXZHUDU
|
7.1 | IC50 | 3 | — | |
OTZHGAAUXLOJFP
|
7.1 | IC50 | 3 | — | |
OYLZIDSUJMGMBF
|
7.1 | IC50 | 3 | — | |
PVDBPOSKQRWTRG
|
7.1 | IC50 | 3 | — | |
TYOPZGWEWQOLHM
|
7.1 | IC50 | 2 | — | |
ULIAHCSBBVNLGS
|
7.1 | IC50 | 3 | — | |
ZBKQSWPCHUEZBL
|
7.1 | IC50 | 3 | — | |
FTHLNVOKHACXIU
|
7.1 | IC50 | 3 | — | |
GWHBOLQUVHIAPZ
|
7.1 | IC50 | 4 | — | |
IPJMGURQBOGYIE
|
7.1 | IC50 | 4 | — | |
ITOTWAQMJPBHEG
|
7.1 | IC50 | 2 | — | |
UBXNLHDUJFHNDS
|
7.1 | IC50 | 3 | — | |
VUWJZAUOMZSUEU
|
7.1 | IC50 | 3 | — | |
ZGCHTGGUXZBHCN
|
7.1 | IC50 | 7 | — | |
BQZRFJLSVVFWBQ
|
7.1 | IC50 | 3 | — | |
LEXSRVMWXAFLMV
|
7.1 | IC50 | 4 | — | |
LEXSRVMWXAFLMV
|
7.1 | IC50 | 3 | — | |
LRWGLQDVNJOJKQ
|
7.1 | IC50 | 3 | — | |
NTLLKKOHPKDCSW
|
7.1 | IC50 | 3 | — | |
PIKWYDHWUKSWAQ
|
7.1 | Kd | 4 | — | |
PMIMBFPXSMELLC
|
7.1 | IC50 | 3 | — | |
UBBQMWGFAITOCR
|
7.1 | IC50 | 2 | — | |
UWHQJIJZHLHELR
|
7.1 | IC50 | 4 | — | |
KGPRTZSROXHRIX
|
7.1 | IC50 | 2 | — |