Target Details
UniProt ACQ15059
Gene SymbolBRD3
Protein NameBromodomain-containing protein 3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF17035 (BET) PF00439 (Bromodomain)
Summary
  • Multi-target molecules 727
  • Clinical molecules 0
  • Avg pChEMBL 7.33
Top Co-occurrence Targets
Active Molecules (727)
InChIKey pChEMBL Type Targets Clinical
JNSLBXJNVHYNNW 10.2 Ki 4
FZWPGKYEENZFAU 10.0 Ki 4
LMLIBNUOIWAJFC 9.5 Kd 9
JIYPVUCBRQNICX 9.3 Kd 7
JNYHQYRTYFSMSQ 9.2 IC50 3
KHQQNXFBTALTQF 9.2 Kd 6
UETQFSCWDMJWMM 9.0 Kd 4
KGERZPVQIRYWRK 9.0 IC50 4
UJARZGSRRXPOTK 8.8 IC50 3
UJARZGSRRXPOTK 8.8 IC50 3
ONTCKBVHGQBHTF 8.7 Ki 3
LZAPXWCSDTYFNB 8.7 IC50 3
AEANZCXROGPSBY 8.7 Kd 6
YPXANNJXRXDMDY 8.6 Ki 3
XYXCJLYWFUGRHO 8.6 Ki 3
FNHHVPPSBFQMEL 8.5 IC50 4
KPWWFNXRLAAREN 8.5 Kd 12
FFQNMMPQMYKTRZ 8.5 Ki 3
WZQLVEPIBAOOGF 8.5 Kd 9
QBWYZTMYCRAFMA 8.4 Ki 3
QFTDPMPFNQAJTK 8.4 Ki 3
DZUPEOBGVVEOJA 8.4 Ki 3
NLHZWVYLQRZHDF 8.4 Ki 3
WOSYEWDDCNUUHT 8.4 IC50 4
PWEXGFMQMFFMNN 8.4 IC50 4
XBGAIUVLEXZQMO 8.4 IC50 4
QUGZCQSQJAUOTO 8.4 Ki 3
HSAHLMIFPRYVEH 8.4 IC50 4
XBGAIUVLEXZQMO 8.4 IC50 4
GCDAPUPAGHUHLH 8.4 IC50 4
VEPYYWIOIMZOLX 8.3 IC50 4
GCDAPUPAGHUHLH 8.3 IC50 4
MFKPAAFGGBINQO 8.3 IC50 4
VYNYPLNNLNISCK 8.3 IC50 4
OEDSFMUSNZDJFD 8.3 IC50 4
RJJDAOYTHRXSGL 8.3 IC50 4
DMSRRTGRIHHJKS 8.3 IC50 4
RKPWYUDCZHEUBU 8.3 IC50 4
UIWJGKYIPQKBHV 8.3 IC50 4
UIWJGKYIPQKBHV 8.3 IC50 4
KMDXJEQFNWVGIH 8.3 Ki 3
RIACYICSJAHABL 8.2 Ki 3
LKEGXJXRNBALBV 8.2 Ki 5
FAWSUKOIROHXAP 8.2 IC50 5
SADKUQHRGVTPSQ 8.2 IC50 4
OJSKWCXPUVTNCF 8.2 IC50 4
WTJMHBMWPMTETL 8.2 IC50 2
YYKYSROKVREYAZ 8.1 IC50 4
MDRXOFSNECSECW 8.1 Ki 4
PQOGZKGXGLHDGS 8.1 Kd 4
2D structure