Target Details
| UniProt AC | Q15047 |
|---|---|
| Gene Symbol | SETDB1 |
| Protein Name | Histone-lysine N-methyltransferase SETDB1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18300 (DUF5604) PF01429 (MBD) PF05033 (Pre-SET) PF00856 (SET) PF18358 (Tudor_4) PF18359 (Tudor_5) |
Summary
- Multi-target molecules 1
- Clinical molecules 0
- Avg pChEMBL 6.68
KEGG Pathways (3)
Top Co-occurrence Targets
- KAT2B 1 shared
Active Molecules (1)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GUFVCUSKHSXTFY
|
6.7 | Kd | 2 | — |