Target Details
| UniProt AC | Q15046 |
|---|---|
| Gene Symbol | KARS1 |
| Protein Name | Lysine--tRNA ligase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00152 (tRNA-synt_2) PF01336 (tRNA_anti-codon) |
Summary
- Multi-target molecules 16
- Clinical molecules 3
- Avg pChEMBL 7.25
KEGG Pathways (1)
Associated Diseases (3)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.1 | IC50 | 408 | — | |
RVIMFNLCTIXVKN
|
8.4 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
8.1 | IC50 | 49 | Yes | |
JMJSTGZRLYHCCI
|
8.1 | IC50 | 5 | — | |
NBGQQTFVANZDGQ
|
8.1 | IC50 | 2 | — | |
SBGMPUIVPOGTGN
|
7.5 | IC50 | 4 | — | |
FQNFLNSVHWCZML
|
7.4 | IC50 | 3 | — | |
VLHKHLQNVJKAHG
|
7.3 | IC50 | 2 | — | |
QMTFEPLRHYDWQT
|
7.1 | IC50 | 2 | — | |
QQVFMNGYKNAGOD
|
6.9 | IC50 | 2 | — | |
OYUDNKFIGXAIRZ
|
6.7 | Ki | 16 | Yes | |
XJSCJPRKDAUMHP
|
6.6 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
6.5 | IC50 | 231 | Yes | |
LPKOEWTZGVUEJF
|
6.2 | IC50 | 3 | — | |
PFQHUUDPALIKDR
|
6.1 | IC50 | 3 | — | |
ZCCPLJOKGAACRT
|
6.1 | Kd | 599 | — |