Target Details
| UniProt AC | Q14832 |
|---|---|
| Gene Symbol | GRM3 |
| Protein Name | Metabotropic glutamate receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00003 (7tm_3) PF01094 (ANF_receptor) PF07562 (NCD3G) |
Summary
- Multi-target molecules 115
- Clinical molecules 0
- Avg pChEMBL 7.29
KEGG Pathways (5)
Active Molecules (115)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QMTVYANBFIIHRR
|
6.5 | IC50 | 2 | — | |
INNYBEXRWKVEPM
|
6.4 | IC50 | 2 | — | |
GZOVEPYOCJWRFC
|
6.4 | Ki | 2 | — | |
XZFMJVJDSYRWDQ
|
6.4 | Ki | 2 | — | |
SUBNOKFHGUEIMG
|
6.4 | IC50 | 2 | — | |
AQCRJOWGCAFEAA
|
6.4 | Ki | 2 | — | |
GZOVEPYOCJWRFC
|
6.4 | Ki | 2 | — | |
LTNANPWTFHLSJB
|
6.3 | IC50 | 2 | — | |
BQVZICWQBFTOJX
|
6.3 | Ki | 2 | — | |
XAWBHQAHNLHFPV
|
6.3 | IC50 | 2 | — | |
BQVZICWQBFTOJX
|
6.2 | Ki | 2 | — | |
ZLLVGXOCXYGTFK
|
6.2 | IC50 | 2 | — | |
YQHUAECMPKPVHE
|
6.2 | IC50 | 2 | — | |
RKBRDSPEJMNTGE
|
6.2 | IC50 | 2 | — | |
MPKHVTSOJQASTK
|
6.1 | IC50 | 2 | — |