Target Details
| UniProt AC | Q14832 |
|---|---|
| Gene Symbol | GRM3 |
| Protein Name | Metabotropic glutamate receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00003 (7tm_3) PF01094 (ANF_receptor) PF07562 (NCD3G) |
Summary
- Multi-target molecules 115
- Clinical molecules 0
- Avg pChEMBL 7.29
KEGG Pathways (5)
Active Molecules (115)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBBCOPQWFRZNNR
|
7.2 | Ki | 2 | — | |
RXZDXHKRDHZRKP
|
7.2 | Ki | 2 | — | |
PZICKINIOPPAGP
|
7.2 | Ki | 2 | — | |
UDWSIQSDTWFRQU
|
7.2 | IC50 | 2 | — | |
NZZMAEBSZGFPBU
|
7.1 | IC50 | 2 | — | |
PZICKINIOPPAGP
|
7.1 | IC50 | 2 | — | |
YKPDUULXXDPIGO
|
7.1 | IC50 | 2 | — | |
KBDQFKQTJBFOTK
|
7.1 | IC50 | 2 | — | |
ZBBCOPQWFRZNNR
|
7.1 | Ki | 2 | — | |
INNYBEXRWKVEPM
|
7.1 | Ki | 2 | — | |
NFWVZCUIJDBXKM
|
7.1 | IC50 | 2 | — | |
ZMUYYXBVNBIBEW
|
7.1 | IC50 | 2 | — | |
QXVMZECHAZYIMZ
|
7.1 | IC50 | 2 | — | |
AVDUGNCTZRCAHH
|
7.0 | Ki | 2 | — | |
JYWMNSYAIWOJGC
|
7.0 | IC50 | 2 | — | |
VTAARTQTOOYTES
|
7.0 | Ki | 2 | — | |
OQCWNVPJUJCZIF
|
7.0 | IC50 | 2 | — | |
NTPXNEQCDPWJQA
|
7.0 | Ki | 2 | — | |
HQTAUDRHEUIJTC
|
6.9 | IC50 | 2 | — | |
XMENKXPGVGTNAZ
|
6.9 | IC50 | 2 | — | |
IGEOMAUWSLBELS
|
6.9 | IC50 | 2 | — | |
YSOWRGMLMZQSBX
|
6.9 | Ki | 2 | — | |
JXTPFQLGVAHAGQ
|
6.8 | IC50 | 2 | — | |
XMDHIHAVEVYYTH
|
6.8 | Ki | 2 | — | |
WNOZOUHFGZKGNT
|
6.8 | IC50 | 2 | — | |
HQTAUDRHEUIJTC
|
6.8 | IC50 | 2 | — | |
YSOWRGMLMZQSBX
|
6.8 | Ki | 2 | — | |
IRMXEKLCWFUGDP
|
6.8 | IC50 | 2 | — | |
HHUBIRLCPJRLDB
|
6.8 | IC50 | 2 | — | |
QSTDCUJNEBAZGO
|
6.8 | IC50 | 2 | — | |
HHUBIRLCPJRLDB
|
6.8 | IC50 | 2 | — | |
HZLKKHXGVUNHPW
|
6.8 | IC50 | 2 | — | |
APZIMAYYQKOWFP
|
6.8 | Ki | 2 | — | |
CNBSEOHDTNDGOV
|
6.8 | IC50 | 2 | — | |
AAZZHVGTJVXBFR
|
6.7 | IC50 | 2 | — | |
GUTXZRKRYGCMAD
|
6.7 | IC50 | 2 | — | |
SGCNJDYPITVHEN
|
6.7 | IC50 | 2 | — | |
MATPZHBYOVDBLI
|
6.7 | Ki | 2 | — | |
MBCWMEYAVJTLQS
|
6.7 | Ki | 2 | — | |
XHHLDXFTATUVFA
|
6.7 | IC50 | 2 | — | |
KPKSEPNXKJWVTO
|
6.6 | IC50 | 2 | — | |
XMENKXPGVGTNAZ
|
6.6 | Ki | 2 | — | |
ASNFTDCKZKHJSW
|
6.6 | Ki | 5 | — | |
XMENKXPGVGTNAZ
|
6.6 | Ki | 2 | — | |
RXZDXHKRDHZRKP
|
6.6 | Ki | 2 | — | |
UBOUWUOIJSJJIT
|
6.6 | IC50 | 2 | — | |
LYTVXCQQTLUEQR
|
6.6 | IC50 | 2 | — | |
LVVJEBBNZXFVDH
|
6.5 | IC50 | 2 | — | |
MHGNPCZGYOTMGN
|
6.5 | Ki | 2 | — | |
JBMRVZCRORVBOW
|
6.5 | IC50 | 2 | — |