Target Details
| UniProt AC | Q14680 |
|---|---|
| Gene Symbol | MELK |
| Protein Name | Maternal embryonic leucine zipper kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF21594 (UBA_MELK) |
Summary
- Multi-target molecules 214
- Clinical molecules 27
- Avg pChEMBL 6.85
Active Molecules (214)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NFMGZVPRGVERNN
|
6.0 | Ki | 44 | — | |
NRGYZNJPCGRCLV
|
6.0 | Ki | 52 | — | |
NRSGWEVTVGZDFC
|
6.0 | Ki | 50 | — | |
PSCJSWRVCKUMSL
|
6.0 | Ki | 35 | — | |
SQXSMLLCDWJNAC
|
6.0 | Ki | 20 | — | |
TZSJMSZEKQGCBI
|
6.0 | Ki | 15 | — | |
VIJBEUTVNBPGIU
|
6.0 | Ki | 19 | — | |
XIOOJUQFJYPVLA
|
6.0 | Ki | 17 | — | |
XKQNBVAZAFAZFL
|
6.0 | IC50 | 6 | — | |
XOVPCPRZRHQFBI
|
6.0 | Ki | 15 | — | |
XYXLUJQBBIBJFV
|
6.0 | Ki | 36 | — | |
YEHCNYAQEBQCCS
|
6.0 | Ki | 74 | — |