Target Details
| UniProt AC | Q14680 |
|---|---|
| Gene Symbol | MELK |
| Protein Name | Maternal embryonic leucine zipper kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF21594 (UBA_MELK) |
Summary
- Multi-target molecules 214
- Clinical molecules 27
- Avg pChEMBL 6.85
Active Molecules (214)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KYACBMRLQMEIAI
|
6.3 | Ki | 30 | — | |
QTQUAHGXBLFSCH
|
6.3 | Ki | 10 | — | |
QXKKPVVOOWBLND
|
6.3 | Ki | 8 | — | |
XSDJOIOVIMPMHD
|
6.3 | Ki | 44 | — | |
ZXLFIHLBHMLHFJ
|
6.3 | Ki | 31 | — | |
ZYTFPHRVOZXPGZ
|
6.3 | Ki | 30 | — | |
FYSDPHKGVBRASN
|
6.3 | IC50 | 4 | — | |
VBYGXNURPHQSPG
|
6.3 | IC50 | 5 | — | |
HHFBDROWDBDFBR
|
6.2 | Kd | 40 | Yes | |
BPNUQXPIQBZCMR
|
6.2 | Kd | 83 | Yes | |
BPNUQXPIQBZCMR
|
6.2 | Ki | 60 | — | |
DZSUJUOJJJCWGG
|
6.2 | Ki | 55 | Yes | |
GQGMUKOYILWOIQ
|
6.2 | Ki | 25 | — | |
HKZKELVPGXJIMW
|
6.2 | Ki | 41 | — | |
KDKUVYLMPJIGKA
|
6.2 | Ki | 91 | Yes | |
KJVWCDAPVMWKLJ
|
6.2 | Ki | 20 | — | |
MCCCQFAOMZMZKE
|
6.2 | Ki | 52 | — | |
MULNSLQVKKUPJN
|
6.2 | Ki | 41 | — | |
MVJMMLFMPWITEJ
|
6.2 | Ki | 110 | — | |
ORUUEFDGYYTXAF
|
6.2 | Ki | 26 | — | |
PBBRWFOVCUAONR
|
6.2 | Ki | 26 | Yes | |
SRROIPFGGDHJCJ
|
6.2 | Ki | 7 | — | |
UUWNXFJBBYAMDT
|
6.2 | Ki | 46 | — | |
XAYDUCQADQTDGX
|
6.2 | Ki | 12 | — | |
XCHWBXBDZRJVDP
|
6.2 | Ki | 51 | — | |
ZGDSBEUMPIMXBM
|
6.2 | Ki | 42 | — | |
LOLPPWBBNUVNQZ
|
6.2 | IC50 | 97 | Yes | |
ZYZUOYYVHYGMDE
|
6.2 | IC50 | 4 | — | |
RQDRHUZBSDGLNX
|
6.1 | IC50 | 2 | — | |
XPLJEFSRINKZLC
|
6.1 | IC50 | 5 | Yes | |
DFMCXVONDDGQIY
|
6.1 | Ki | 66 | — | |
GUMBHNMWKMFKRT
|
6.1 | Ki | 23 | — | |
JCFJQIHDZHHMQT
|
6.1 | Ki | 42 | — | |
JJTYLBBKGQOISV
|
6.1 | Ki | 15 | — | |
LGHBDVLAHHANMX
|
6.1 | Ki | 53 | — | |
MQRDVGBWWVWMEN
|
6.1 | Ki | 47 | — | |
OLVBAUVSICCWEJ
|
6.1 | Ki | 39 | — | |
UMYBAQLXZPEUQW
|
6.1 | Ki | 15 | — | |
VSPFURGQAYMVAN
|
6.1 | Ki | 17 | — | |
XKFTZKGMDDZMJI
|
6.1 | Ki | 56 | — | |
XLFYOIVELARSKP
|
6.1 | Ki | 33 | — | |
ODPGGGTTYSGTGO
|
6.1 | Kd | 153 | — | |
AILRADAXUVEEIR
|
6.0 | IC50 | 75 | — | |
FWLMVFUGMHIOAA
|
6.0 | Kd | 26 | — | |
KGPGFQWBCSZGEL
|
6.0 | Kd | 59 | Yes | |
UKBGBACORPRCGG
|
6.0 | IC50 | 17 | — | |
FLBNLJLONKAPLR
|
6.0 | Kd | 31 | — | |
BZFGDXJGWSIYQP
|
6.0 | Ki | 9 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KCKXYZOBGBJZEG
|
6.0 | Ki | 36 | — |