Target Details
| UniProt AC | Q14680 |
|---|---|
| Gene Symbol | MELK |
| Protein Name | Maternal embryonic leucine zipper kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF21594 (UBA_MELK) |
Summary
- Multi-target molecules 214
- Clinical molecules 27
- Avg pChEMBL 6.85
Active Molecules (214)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SGZZQKMOFHIDKW
|
6.7 | IC50 | 13 | — | |
YAJKTHRIWKTLDH
|
6.7 | IC50 | 2 | — | |
AXTAPYRUEKNRBA
|
6.6 | Kd | 24 | — | |
GCIKSSRWRFVXBI
|
6.6 | Kd | 109 | Yes | |
GHPFSYCYZJKVDZ
|
6.6 | Ki | 18 | Yes | |
GXJSLIOOPZRPEV
|
6.6 | Ki | 34 | — | |
LRZYYIZFBXFSJB
|
6.6 | Ki | 69 | — | |
PTVPBWWDGZSEAF
|
6.6 | Ki | 63 | — | |
VXYDJXMHISGSDA
|
6.6 | Ki | 59 | — | |
WKEYMNLZBZKLOG
|
6.6 | Ki | 14 | — | |
WPHKIQPVPYJNAX
|
6.6 | Ki | 81 | — | |
XQVVPGYIWAGRNI
|
6.6 | Ki | 19 | — | |
KZVIZFHCMVWFNT
|
6.6 | IC50 | 7 | — | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 91 | Yes | |
CXQHYVUVSFXTMY
|
6.5 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.5 | Kd | 149 | — | |
CLEGDJQQHUTCOW
|
6.5 | Ki | 43 | — | |
CYLGCMABIBXHIQ
|
6.5 | Ki | 16 | — | |
MASJMHFQMYAPJR
|
6.5 | Ki | 41 | — | |
QKPLUKMJEKRAJD
|
6.5 | Ki | 30 | Yes | |
RIBBPSYZBQQTQC
|
6.5 | Ki | 15 | — | |
UYJNQQDJUOUFQJ
|
6.5 | Ki | 68 | — | |
VUHZDNOPEVGHEO
|
6.5 | Ki | 29 | — | |
YWTBGJGMTBHQTM
|
6.5 | Ki | 65 | — | |
VNDWQCSOSCCWIP
|
6.5 | IC50 | 39 | Yes | |
CTNPALGJUAXMMC
|
6.5 | Kd | 151 | — | |
XDJCLCLBSGGNKS
|
6.5 | IC50 | 21 | — | |
WINHZLLDWRZWRT
|
6.5 | Kd | 201 | Yes | |
AOBLBPWPSKBHSI
|
6.4 | Ki | 55 | — | |
FAYAUAZLLLJJGH
|
6.4 | Ki | 36 | Yes | |
FDVSOQRNTAPCHB
|
6.4 | Ki | 40 | — | |
HJYHJYGXRBYDIG
|
6.4 | Ki | 23 | — | |
HRZOUBQYVUXBNS
|
6.4 | Ki | 38 | — | |
KRIUNPBAQZGFQA
|
6.4 | Ki | 76 | — | |
LRLDYTTWQIFWBD
|
6.4 | Ki | 25 | — | |
MMFBBQQGBVPLQQ
|
6.4 | Ki | 13 | — | |
PCQMERRARZKTPW
|
6.4 | Ki | 68 | — | |
PDBPUXLUVDSLML
|
6.4 | Ki | 14 | — | |
QNUKRWAIZMBVCU
|
6.4 | Ki | 46 | — | |
QTHCAAFKVUWAFI
|
6.4 | IC50 | 23 | — | |
RJZDECGDCKOHBV
|
6.4 | Ki | 70 | — | |
UDFDIIVNIYWXDM
|
6.4 | Ki | 74 | — | |
UZFPGFONVYFSRR
|
6.4 | Ki | 16 | — | |
XFWUTMHVDGPWLH
|
6.4 | Ki | 75 | — | |
XMFUGSRATNLPRM
|
6.4 | Ki | 19 | — | |
YACXOXQTGJXYNX
|
6.4 | Ki | 11 | — | |
ZGZVRPRSFXRGCF
|
6.4 | Ki | 76 | — | |
GDYZFFBMSBDTAA
|
6.3 | Ki | 60 | — | |
HEUSUIRCBWROMH
|
6.3 | Ki | 64 | — |