Target Details
| UniProt AC | Q14680 |
|---|---|
| Gene Symbol | MELK |
| Protein Name | Maternal embryonic leucine zipper kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF21594 (UBA_MELK) |
Summary
- Multi-target molecules 214
- Clinical molecules 27
- Avg pChEMBL 6.85
Active Molecules (214)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AYCPARAPKDAOEN
|
7.2 | Kd | 73 | — | |
OFIFLUFVENTCNZ
|
7.2 | IC50 | 11 | — | |
PRRYQINUAIQTFJ
|
7.2 | Ki | 11 | — | |
UTQPKPHUIMHAAN
|
7.2 | Ki | 22 | — | |
XJSFDMGICAWQFS
|
7.2 | Ki | 60 | — | |
IABDKYMGRMDGMM
|
7.1 | Ki | 10 | — | |
KWRXWPRFIUJQBP
|
7.1 | Ki | 25 | — | |
KXPWWMPXNUOYOH
|
7.1 | Ki | 24 | — | |
MZDKLVOWGIOKTN
|
7.1 | Ki | 80 | — | |
NJPWCTYVEJIQBM
|
7.1 | Ki | 72 | — | |
WUBHCQHBUVGGRX
|
7.1 | Ki | 11 | — | |
WYOMXSAYYXBPMN
|
7.1 | Ki | 24 | — | |
KOZFSFOOLUUIGY
|
7.1 | Kd | 88 | Yes | |
MSWOWUREQODTRO
|
7.0 | IC50 | 11 | — | |
GQLWKGVBOIYMTN
|
7.0 | Ki | 35 | — | |
OWRXHGAFWZFFCW
|
7.0 | Ki | 113 | — | |
QONPPIZSNSSCSK
|
7.0 | Ki | 45 | Yes | |
QQWUGDVOUVUTOY
|
7.0 | Kd | 231 | Yes | |
XOOAAYRIVATZNM
|
7.0 | Ki | 55 | — | |
XPHWIERLJBFPFV
|
7.0 | Ki | 69 | — | |
ACPOUJIDANTYHO
|
7.0 | IC50 | 17 | Yes | |
ADMFLILDQJSEIK
|
6.9 | Ki | 72 | — | |
BEJCLDKQCNVTQR
|
6.9 | Ki | 16 | — | |
CRKQBJZCCHKEGI
|
6.9 | Ki | 20 | — | |
DKSNLQYRZJKYOC
|
6.9 | Ki | 51 | — | |
GSXRCPJTNIGKSZ
|
6.9 | Ki | 43 | — | |
ZWVZORIKUNOTCS
|
6.9 | Ki | 69 | — | |
DUKJABPGWUISRC
|
6.8 | IC50 | 10 | — | |
FTIAKTLRFKSDFR
|
6.8 | Ki | 10 | Yes | |
JSKUWFIZUALZLX
|
6.8 | Ki | 33 | — | |
KAZJIBCOYQRDGG
|
6.8 | Ki | 16 | — | |
OUSFTKFNBAZUKL
|
6.8 | Ki | 58 | Yes | |
SFPWNTQWFFNJIH
|
6.8 | Ki | 48 | — | |
WZISGNDZZPSYRP
|
6.8 | Ki | 20 | — | |
MFAQYJIYDMLAIM
|
6.8 | Kd | 130 | Yes | |
AZTMYWWWILJAKW
|
6.7 | Ki | 16 | Yes | |
CHTMRWQLNNRRFJ
|
6.7 | Ki | 70 | — | |
GXTJETQFYHZHNB
|
6.7 | IC50 | 2 | — | |
HHSVICUMCOBRPT
|
6.7 | Ki | 33 | — | |
HSKVRPZJBMXFDX
|
6.7 | Ki | 20 | — | |
JBJIKUXUKSADFV
|
6.7 | IC50 | 3 | — | |
MIKAKZKNMYZLDX
|
6.7 | Ki | 42 | — | |
OETCTXGISYWYMV
|
6.7 | Ki | 7 | — | |
OUJZYQBEFNDJQN
|
6.7 | Ki | 71 | — | |
RYYNGWLOYLRZLK
|
6.7 | Ki | 104 | — | |
WLTSTDGGFCQWTK
|
6.7 | IC50 | 3 | — | |
WVFWTUJEHMVUBG
|
6.7 | Ki | 25 | — | |
XYZNKCSDQRKAFR
|
6.7 | Ki | 53 | — | |
YYLKKYCXAOBSRM
|
6.7 | Kd | 191 | — | |
GLDSKRNGVVYJAB
|
6.7 | IC50 | 16 | — |