Target Details
| UniProt AC | Q14680 |
|---|---|
| Gene Symbol | MELK |
| Protein Name | Maternal embryonic leucine zipper kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF21594 (UBA_MELK) |
Summary
- Multi-target molecules 214
- Clinical molecules 27
- Avg pChEMBL 6.85
Active Molecules (214)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.5 | Ki | 118 | — | |
RFBPWKMQWSIPEO
|
9.0 | Ki | 28 | — | |
DKZYXHCYPUVGAF
|
9.0 | IC50 | 112 | — | |
PLHUMPJXRHMFFR
|
8.9 | Ki | 28 | — | |
ZKLJKKASNXVQBZ
|
8.9 | Ki | 27 | — | |
HKSZLNNOFSGOKW
|
8.9 | IC50 | 408 | — | |
FCLPVPNWFDOVKL
|
8.9 | IC50 | 11 | — | |
DQPYZHUAILXFJI
|
8.8 | Ki | 27 | — | |
KHGPYYFCIAISBU
|
8.8 | Ki | 31 | — | |
NOMBUNHXDWBICV
|
8.7 | IC50 | 11 | — | |
XNWKXXIGSPPPBH
|
8.7 | Ki | 31 | — | |
HYUGTGGDEAGXJP
|
8.6 | IC50 | 11 | — | |
WGWCRXQUBYJTRA
|
8.5 | IC50 | 11 | — | |
WDARYLSSWBWVCU
|
8.5 | Ki | 49 | — | |
XUFLBSMTYMFOQH
|
8.5 | Ki | 43 | — | |
CFIBXVQLBVNOHW
|
8.4 | Ki | 64 | — | |
ACSYKUPGCXYRRO
|
8.3 | Ki | 26 | — | |
BSFNGHCTZDCQBF
|
8.3 | Ki | 93 | — | |
FUMCKNCUEAQHCV
|
8.3 | Ki | 103 | — | |
PUYIXDDMOUMMRR
|
8.3 | Ki | 27 | — | |
WMWHVTDZNIVNIE
|
8.3 | IC50 | 9 | — | |
WMWHVTDZNIVNIE
|
8.3 | IC50 | 9 | — | |
GCYXEGSPUDSZJY
|
8.2 | Ki | 82 | — | |
UYGYYOIUVFMGKQ
|
8.2 | Ki | 30 | — | |
NBMVLIXNQOYMFB
|
8.1 | Kd | 2 | — | |
KQVNWJXQFRWTDU
|
8.0 | Kd | 2 | — | |
GQQAKEHCSMJAKS
|
7.9 | Kd | 2 | — | |
SRKBDTMNOSQJFR
|
7.9 | Kd | 2 | — | |
ZCCPLJOKGAACRT
|
7.8 | Kd | 599 | — | |
HSMUWLLZAZCLHF
|
7.8 | Ki | 25 | — | |
UMTWTCVTRDYHQQ
|
7.8 | Ki | 56 | — | |
FTDWSWREBGYXDZ
|
7.7 | IC50 | 10 | — | |
LCHCSKHPVCDXAU
|
7.7 | Ki | 30 | — | |
LACOMQAWPSFXQC
|
7.6 | Ki | 27 | — | |
SMRWVXLSRJWVBF
|
7.6 | Ki | 25 | — | |
PBACTZXZNFJQGT
|
7.6 | IC50 | 4 | — | |
UIARLYUEJFELEN
|
7.6 | Kd | 289 | Yes | |
JFKIXRTUZAZONT
|
7.5 | Ki | 6 | — | |
PIQCTGMSNWUMAF
|
7.5 | Ki | 137 | Yes | |
HKSZLNNOFSGOKW
|
7.5 | Kd | 213 | — | |
GMZCYCKIXQZORP
|
7.4 | IC50 | 6 | — | |
FLEAYYMORDPWAJ
|
7.4 | Ki | 90 | — | |
RWKDVIAVTRRJIR
|
7.4 | Ki | 23 | — | |
OSVUGUHRKMMBSE
|
7.4 | Kd | 170 | — | |
XZXHXSATPCNXJR
|
7.4 | IC50 | 165 | Yes | |
CKVWQORGCCEYHS
|
7.3 | Ki | 50 | — | |
NLDZIKOJZCTRAZ
|
7.3 | Ki | 5 | — | |
NXSJMRCTGYTSTK
|
7.3 | Kd | 200 | — | |
QATMNAAQTUISJK
|
7.3 | Ki | 13 | — | |
XZONYYFHQICDAM
|
7.3 | Ki | 19 | — |