Target Details
| UniProt AC | Q14676 |
|---|---|
| Gene Symbol | MDC1 |
| Protein Name | Mediator of DNA damage checkpoint protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16589 (BRCT_2) PF00498 (FHA) PF16770 (RTT107_BRCT_5) |
Summary
- Multi-target molecules 6
- Clinical molecules 0
- Avg pChEMBL 7.77
Active Molecules (6)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IXZOHGPZAQLIBH
|
8.7 | IC50 | 8 | — | |
IXZOHGPZAQLIBH
|
8.6 | IC50 | 6 | — | |
IXZOHGPZAQLIBH
|
7.9 | IC50 | 6 | — | |
UVSMNLNDYGZFPF
|
7.5 | IC50 | 7 | — | |
RSNPAKAFCAAMBH
|
7.2 | IC50 | 8 | — | |
GOTYRUGSSMKFNF
|
6.7 | IC50 | 6 | — |