Target Details
| UniProt AC | Q14654 |
|---|---|
| Gene Symbol | KCNJ11 |
| Protein Name | ATP-sensitive inward rectifier potassium channel 11 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01007 (IRK) PF17655 (IRK_C) |
Summary
- Multi-target molecules 29
- Clinical molecules 0
- Avg pChEMBL 6.66
KEGG Pathways (3)
Associated Diseases (5)
Active Molecules (29)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IYANXPKCSGLCRO
|
8.5 | IC50 | 2 | — | |
HKZNADVVGXKQDL
|
7.6 | Ki | 2 | — | |
PSCXSSQRAGJZST
|
7.1 | Ki | 2 | — | |
LVEDGSIMCSQNNX
|
7.1 | IC50 | 4 | — | |
XUSQKHZVTSWKMN
|
7.1 | IC50 | 2 | — | |
PGYDRGZVXVVZQC
|
7.0 | Ki | 2 | — | |
TVZCRIROJQEVOT
|
7.0 | IC50 | 4 | — | |
ZHGCRRVSTOTYSM
|
6.9 | IC50 | 2 | — | |
CBVDKJDKOREVOE
|
6.9 | IC50 | 4 | — | |
ZNNLBTZKUZBEKO
|
6.9 | IC50 | 5 | — | |
NMMSLDYACYCEND
|
6.8 | Ki | 2 | — | |
ZSVQNUGFXADOQI
|
6.7 | IC50 | 2 | — | |
HEOGMAJPFJKOND
|
6.6 | IC50 | 2 | — | |
KYSFUHHFTIGRJN
|
6.5 | IC50 | 2 | — | |
IVVNZDGDKPTYHK
|
6.5 | Ki | 2 | — | |
NDBOSDQLHXHDSC
|
6.5 | IC50 | 2 | — | |
USMNFLTXHACNKB
|
6.5 | Ki | 2 | — | |
PXUHSBKGJFYMON
|
6.4 | IC50 | 4 | — | |
KGNPNVWVGXSHJT
|
6.3 | IC50 | 2 | — | |
LJLXQHHFAKVTNP
|
6.3 | IC50 | 4 | — | |
LTKRZCMBXQFJLK
|
6.3 | IC50 | 4 | — | |
VUTFALFOMNJMQI
|
6.3 | Ki | 2 | — | |
TVZCRIROJQEVOT
|
6.3 | IC50 | 4 | — | |
GNVWYNKNTYVESS
|
6.3 | IC50 | 4 | — | |
XKQUHPOBIFXEAQ
|
6.2 | IC50 | 4 | — | |
KGNPNVWVGXSHJT
|
6.2 | IC50 | 2 | — | |
BNIZYODSEJZOIY
|
6.2 | Ki | 2 | — | |
DYMOQRBZQBQYDN
|
6.1 | IC50 | 4 | — | |
XIPHANJESHAHDZ
|
6.1 | IC50 | 4 | — |