Target Details
| UniProt AC | Q14524 |
|---|---|
| Gene Symbol | SCN5A |
| Protein Name | Sodium channel protein type 5 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 683
- Clinical molecules 2
- Avg pChEMBL 7.49
KEGG Pathways (2)
Associated Diseases (8)
Active Molecules (683)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WBUKUXXILSESLB
|
7.5 | IC50 | 3 | — | |
CQNROXJZTLLINO
|
7.5 | IC50 | 2 | — | |
JAUQXVXTUFWMRU
|
7.5 | IC50 | 2 | — | |
KUEJLJXMCCPJMA
|
7.5 | IC50 | 2 | — | |
NEGWWOJFNIDTET
|
7.5 | IC50 | 2 | — | |
ZECJEHQTOHGKFP
|
7.5 | IC50 | 2 | — | |
JZQURVBEWWCEHW
|
7.5 | IC50 | 2 | — | |
RUJWRSKJYRGFJT
|
7.5 | IC50 | 2 | — | |
UOEUNSIONXILJG
|
7.5 | IC50 | 2 | — | |
AQCJPKSGNJCPEK
|
7.5 | IC50 | 2 | — | |
CIXVIWMKNATLIZ
|
7.5 | IC50 | 3 | — | |
GCVAXVXEWOIGNP
|
7.5 | IC50 | 2 | — | |
AQCJPKSGNJCPEK
|
7.5 | IC50 | 2 | — | |
CQMGOVSDXNMSHT
|
7.5 | IC50 | 2 | — | |
ALEKFWIWCIMWKG
|
7.5 | IC50 | 3 | — | |
KRNHAUPCKRIYSK
|
7.5 | IC50 | 3 | — | |
OZAYOHJGXLWETR
|
7.5 | IC50 | 2 | — | |
BKXDCUIYPNHSRV
|
7.5 | IC50 | 2 | — | |
WNMVVEMAMGPLOA
|
7.5 | IC50 | 2 | — | |
PXIOSRRDENCWDU
|
7.5 | IC50 | 2 | — | |
GFVCFLPKZWOAQW
|
7.5 | IC50 | 2 | — | |
NVDJRUZWJVKEIQ
|
7.5 | IC50 | 3 | — | |
ROVKLDKSHHGRMO
|
7.5 | IC50 | 2 | — | |
KHAPUVAAGNEHQW
|
7.4 | IC50 | 2 | — | |
SDFWLGIHLRLHLP
|
7.4 | IC50 | 3 | — | |
IRQCHFVTFWRVCS
|
7.4 | IC50 | 2 | — | |
ISZSRLNGUGMFAI
|
7.4 | IC50 | 2 | — | |
YSAHUUYUAWFVKI
|
7.4 | IC50 | 2 | — | |
XMVKPHXYJPWNBI
|
7.4 | IC50 | 2 | — | |
GMQMLOXLGZOQFR
|
7.4 | IC50 | 2 | — | |
BJWSTFAHQAKCBG
|
7.4 | IC50 | 2 | — | |
DEYOMPPOEBPYPT
|
7.4 | IC50 | 3 | — | |
HAYGNNHVUSBUBN
|
7.4 | IC50 | 3 | — | |
INMXDYHKDXGDPC
|
7.4 | IC50 | 2 | — | |
KGXDTVHRHKTTQK
|
7.4 | IC50 | 2 | — | |
MWSVLDOKXAVVNZ
|
7.4 | IC50 | 3 | — | |
NBEBBBQDSOMUAC
|
7.4 | IC50 | 2 | — | |
WDDGGSNPHYNGMF
|
7.4 | IC50 | 2 | — | |
DRNSHRBRTNNNRM
|
7.4 | IC50 | 2 | — | |
JNRFJFSNMOLYBU
|
7.4 | IC50 | 2 | — | |
GQIRJGCLEQYBML
|
7.4 | IC50 | 3 | — | |
SOMCQNIHPYFNEM
|
7.4 | IC50 | 2 | — | |
SQHCXAPOOMTODU
|
7.4 | IC50 | 2 | — | |
GFUJFOMKFGBYEO
|
7.4 | IC50 | 2 | — | |
OAHIMSPLYGQQRM
|
7.4 | IC50 | 2 | — | |
XTZUOCSNLORVFV
|
7.4 | IC50 | 2 | — | |
LIFZJXOUFVMMPM
|
7.4 | IC50 | 2 | — | |
DKLFTDOPHVNBBI
|
7.3 | IC50 | 3 | — | |
DCSIWUFDXHSLND
|
7.3 | IC50 | 2 | — | |
DVIIENUECJXHTK
|
7.3 | IC50 | 2 | — |