Target Details
| UniProt AC | Q14524 |
|---|---|
| Gene Symbol | SCN5A |
| Protein Name | Sodium channel protein type 5 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 683
- Clinical molecules 2
- Avg pChEMBL 7.49
KEGG Pathways (2)
Associated Diseases (8)
Active Molecules (683)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WXFLUTLJETXITM
|
7.8 | IC50 | 2 | — | |
GCVLCXXOZKDWKX
|
7.8 | IC50 | 2 | — | |
OCNOGKDYKRVBCZ
|
7.8 | IC50 | 3 | — | |
SDFWLGIHLRLHLP
|
7.8 | IC50 | 3 | — | |
SJCKDZDWCFXPHT
|
7.8 | IC50 | 2 | — | |
QJNYOQCRJJMAOZ
|
7.8 | IC50 | 3 | — | |
QEQUMUCQZCHHBH
|
7.8 | IC50 | 2 | — | |
CQOUGURSFKSLMF
|
7.8 | IC50 | 2 | — | |
FNXPIKCUIQCFFD
|
7.8 | IC50 | 2 | — | |
YJHJXTTXJRZIOQ
|
7.8 | IC50 | 2 | — | |
HBNLKZBNOCBHIO
|
7.8 | IC50 | 2 | — | |
AUMPIEINVCBDOI
|
7.8 | IC50 | 2 | — | |
GCVLCXXOZKDWKX
|
7.8 | IC50 | 2 | — | |
NDHYFBZFYCXQJV
|
7.8 | IC50 | 2 | — | |
OGXYRLBTADEONS
|
7.8 | IC50 | 2 | — | |
VDOLFGHRDHGMCS
|
7.8 | IC50 | 2 | — | |
VQBGPJJILMRFBJ
|
7.8 | IC50 | 2 | — | |
BJUGCVMDGAASCX
|
7.7 | IC50 | 2 | — | |
KPHLEZXDKXIWFG
|
7.7 | IC50 | 2 | — | |
RAMYNPHHIXANPH
|
7.7 | IC50 | 2 | — | |
YSAHUUYUAWFVKI
|
7.7 | IC50 | 2 | — | |
RCAXTKUIFXSBJK
|
7.7 | IC50 | 2 | — | |
BJUGCVMDGAASCX
|
7.7 | IC50 | 2 | — | |
DLVHLOHKEQWDBO
|
7.7 | IC50 | 2 | — | |
PNUXVRFTINUPJH
|
7.7 | IC50 | 3 | — | |
SFDBYELGYJKPAZ
|
7.7 | IC50 | 2 | — | |
SREGSGWKZFYIDY
|
7.7 | IC50 | 3 | — | |
CQNROXJZTLLINO
|
7.7 | IC50 | 2 | — | |
OVHKFCHMFRAKJC
|
7.7 | IC50 | 2 | — | |
BSHIKYSNYVZEIY
|
7.7 | IC50 | 2 | — | |
HBNLKZBNOCBHIO
|
7.7 | IC50 | 2 | — | |
GHTDSDKXPCEXRT
|
7.7 | IC50 | 2 | — | |
GQIRJGCLEQYBML
|
7.7 | IC50 | 3 | — | |
JBECBHNSFAXSII
|
7.7 | IC50 | 2 | — | |
UVPFUHLMKQGWHA
|
7.7 | IC50 | 2 | — | |
DLVHLOHKEQWDBO
|
7.7 | IC50 | 2 | — | |
TXWCGOIFALQYHQ
|
7.7 | IC50 | 2 | — | |
GZNHRVQDDAHXKN
|
7.6 | IC50 | 2 | — | |
HFUQIJGZENHTPZ
|
7.6 | IC50 | 2 | — | |
QQSAJPXJGRDAMG
|
7.6 | IC50 | 2 | — | |
UIBQRFPOJVQWAL
|
7.6 | IC50 | 2 | — | |
KNWMNXSIMFAJLJ
|
7.6 | IC50 | 2 | — | |
PVIGPMARFARWPP
|
7.6 | IC50 | 2 | — | |
WEOKXLHSGGJADC
|
7.6 | IC50 | 2 | — | |
UAQLRELQQBERST
|
7.6 | IC50 | 2 | — | |
XONVETJGMAXMDQ
|
7.6 | IC50 | 2 | — | |
FCTRCSDOQULOAY
|
7.6 | IC50 | 2 | — | |
OXIBUPUBHKVZRW
|
7.6 | IC50 | 2 | — | |
MUSMJSIOKVJKDY
|
7.6 | IC50 | 2 | — | |
WOCJXCJKUKAOGM
|
7.5 | IC50 | 2 | — |