Target Details
| UniProt AC | Q14524 |
|---|---|
| Gene Symbol | SCN5A |
| Protein Name | Sodium channel protein type 5 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 683
- Clinical molecules 2
- Avg pChEMBL 7.49
KEGG Pathways (2)
Associated Diseases (8)
Active Molecules (683)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LLQGWDGJRDPIES
|
8.0 | IC50 | 2 | — | |
ODRKYAAJDAGRKU
|
8.0 | IC50 | 2 | — | |
PNUVCZLZKVPMSF
|
8.0 | IC50 | 2 | — | |
QDFFMRBOHNMZAT
|
8.0 | IC50 | 2 | — | |
QWGWIALEIALNJD
|
8.0 | IC50 | 2 | — | |
XONVETJGMAXMDQ
|
8.0 | IC50 | 2 | — | |
DJSYVSUYNVQSCR
|
8.0 | IC50 | 2 | — | |
QMOLJXRAMAPQPQ
|
8.0 | IC50 | 2 | — | |
SAECGYZACNUJAE
|
8.0 | IC50 | 2 | — | |
AHLYPDZHXOGAAC
|
8.0 | IC50 | 2 | — | |
HTYPEQFLNSKYPG
|
8.0 | IC50 | 2 | — | |
KYELVWPATFRSJQ
|
8.0 | IC50 | 2 | — | |
MVEPDUKIVTZGJC
|
8.0 | IC50 | 2 | — | |
TWTAHZZUGXMXLY
|
8.0 | IC50 | 2 | — | |
VUSBGJHOMNTZQY
|
8.0 | IC50 | 2 | — | |
WHVCUTYOIICUIK
|
8.0 | IC50 | 2 | — | |
ZYSCOUXLBXGGIM
|
8.0 | IC50 | 9 | — | |
FQIILMZKICAGTI
|
8.0 | IC50 | 2 | — | |
MDLDNPVKBYFOTI
|
8.0 | IC50 | 2 | — | |
PIWYVIVUOSLKSX
|
8.0 | IC50 | 2 | — | |
XIMWGAYQBHYLSU
|
8.0 | IC50 | 2 | — | |
KSGFLCHXWLJABA
|
7.9 | IC50 | 2 | — | |
SDJQJNMYRSLYAF
|
7.9 | IC50 | 2 | — | |
ZEOCEVMDPZIHPM
|
7.9 | IC50 | 2 | — | |
JZQURVBEWWCEHW
|
7.9 | IC50 | 2 | — | |
MMUQDMQKMOLLET
|
7.9 | IC50 | 2 | — | |
QMIHBNPMTMLUMI
|
7.9 | IC50 | 3 | — | |
TWTAHZZUGXMXLY
|
7.9 | IC50 | 2 | — | |
UHNGVVPJTQLYJP
|
7.9 | IC50 | 2 | — | |
GOERNEVEZCWLDT
|
7.9 | IC50 | 2 | — | |
FKPOFESGNHGZMW
|
7.9 | IC50 | 2 | — | |
KDVYWGKDSHINDP
|
7.9 | IC50 | 2 | — | |
NEWRVLYCADPFOU
|
7.9 | IC50 | 2 | — | |
HBYPLMPPHBGEDI
|
7.9 | IC50 | 2 | — | |
IRFMFQQIANLALO
|
7.9 | IC50 | 2 | — | |
PCWUHIYHTMODIL
|
7.9 | IC50 | 2 | — | |
SCZYLEWDHRXONF
|
7.9 | IC50 | 2 | — | |
IFEGKGXITIRTCE
|
7.9 | IC50 | 2 | — | |
PLZANXMHAHDQEY
|
7.9 | IC50 | 2 | — | |
DUTBELDPUMKBDW
|
7.8 | IC50 | 2 | — | |
NZLJRXFUYNPRME
|
7.8 | IC50 | 2 | — | |
RHLSSDADJRDXLU
|
7.8 | IC50 | 2 | — | |
WHVCUTYOIICUIK
|
7.8 | IC50 | 2 | — | |
ZHOVMQJWRQDRFQ
|
7.8 | IC50 | 2 | — | |
GFVCFLPKZWOAQW
|
7.8 | IC50 | 2 | — | |
KYERELZTVNAFJL
|
7.8 | IC50 | 2 | — | |
VLIGDXLMKUKWJZ
|
7.8 | IC50 | 2 | — | |
CDWKRWXCVDRSRN
|
7.8 | IC50 | 2 | — | |
GIYHIVFXKAMIDY
|
7.8 | IC50 | 2 | — | |
OXLXEJBCNSQASQ
|
7.8 | IC50 | 2 | — |