Target Details
| UniProt AC | Q14524 |
|---|---|
| Gene Symbol | SCN5A |
| Protein Name | Sodium channel protein type 5 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 683
- Clinical molecules 2
- Avg pChEMBL 7.49
KEGG Pathways (2)
Associated Diseases (8)
Active Molecules (683)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KHAPUVAAGNEHQW
|
8.3 | IC50 | 2 | — | |
QQRDUMOOLIZBOV
|
8.3 | IC50 | 2 | — | |
RJZUNWGDQAGCHL
|
8.3 | IC50 | 2 | — | |
XDAKREHNKKKEAQ
|
8.3 | IC50 | 2 | — | |
ZVROQFJWLWNYPQ
|
8.3 | IC50 | 2 | — | |
KTQITWVXYXCIPI
|
8.3 | IC50 | 2 | — | |
WWPICVXQOKPCAZ
|
8.3 | IC50 | 2 | — | |
YSEGGAVVNUBFOR
|
8.3 | IC50 | 2 | — | |
BHNHPSMLNIXZEA
|
8.3 | IC50 | 2 | — | |
FUFQYXJEKPAYHJ
|
8.3 | IC50 | 2 | — | |
ICDZOMMZQJGZGT
|
8.3 | IC50 | 2 | — | |
LNZNUXVENBAPOZ
|
8.3 | IC50 | 2 | — | |
PBBRTUUYKGXANR
|
8.3 | IC50 | 2 | — | |
PRCIGHMFXRYAIG
|
8.3 | IC50 | 3 | — | |
QWKZXVRTHGUGEI
|
8.3 | IC50 | 2 | — | |
UUYBPWNOSQSJHQ
|
8.3 | IC50 | 2 | — | |
YEUQOLDVWRDBED
|
8.3 | IC50 | 2 | — | |
ZVROQFJWLWNYPQ
|
8.3 | IC50 | 2 | — | |
BVOXFWHQWQANHR
|
8.3 | IC50 | 2 | — | |
BYPCGZJBGJSUGQ
|
8.3 | IC50 | 2 | — | |
IDJPUZREEMOMJC
|
8.3 | IC50 | 2 | — | |
IKDXHRATCNECAM
|
8.3 | IC50 | 2 | — | |
JEZPXQKQZQRRMC
|
8.3 | IC50 | 2 | — | |
KWAURGCHFYCYPQ
|
8.2 | IC50 | 4 | — | |
LKWRNZBTPSCWJT
|
8.2 | IC50 | 3 | — | |
MQBAFWXBAHSNIS
|
8.2 | IC50 | 2 | — | |
DDOIQOFHDMJGBP
|
8.2 | IC50 | 2 | — | |
DPKBSJIWLASXHR
|
8.2 | IC50 | 2 | — | |
GNHOWCLPSIXZMF
|
8.2 | IC50 | 2 | — | |
HDQYQOWHBKXUCR
|
8.2 | IC50 | 2 | — | |
KRRQPHNWSHNADQ
|
8.2 | IC50 | 2 | — | |
QFOGEZLLIKAJNO
|
8.2 | IC50 | 2 | — | |
VQJZDKCEVLXOTH
|
8.2 | IC50 | 2 | — | |
OCUQANFWZAMQKA
|
8.2 | IC50 | 2 | — | |
DQSHMENCHXKIOD
|
8.2 | IC50 | 2 | — | |
FLRIBHCWDYEBHH
|
8.2 | IC50 | 2 | — | |
HJRAXXVKFXITKI
|
8.2 | IC50 | 2 | — | |
HRRHRSSCWYTCBS
|
8.2 | IC50 | 3 | — | |
IKGSSFBIKHWXLY
|
8.2 | IC50 | 2 | — | |
KMXYAYHLGANJIA
|
8.2 | IC50 | 2 | — | |
WFIDFECCLBIDBW
|
8.2 | IC50 | 2 | — | |
ABFJGJYHHOCPJV
|
8.2 | IC50 | 2 | — | |
BRVBRZABHLGTRI
|
8.2 | IC50 | 2 | — | |
MKTFWIFFQBKEFV
|
8.2 | IC50 | 2 | — | |
NQDCRCJMPKRFBR
|
8.2 | IC50 | 2 | — | |
QJCLEBMUIYIWPM
|
8.2 | IC50 | 2 | — | |
BBTLYGRMWYLRGJ
|
8.2 | IC50 | 2 | — | |
LRXJCQGUTGFUKQ
|
8.2 | IC50 | 2 | — | |
VONKMVXDHIRYQE
|
8.2 | IC50 | 2 | — | |
WJLZKECJHILDNE
|
8.2 | IC50 | 2 | — |