Target Details
| UniProt AC | Q14524 |
|---|---|
| Gene Symbol | SCN5A |
| Protein Name | Sodium channel protein type 5 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 683
- Clinical molecules 2
- Avg pChEMBL 7.49
KEGG Pathways (2)
Associated Diseases (8)
Active Molecules (683)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JZQURVBEWWCEHW
|
8.4 | IC50 | 2 | — | |
KYBPOTYVFWNSGS
|
8.4 | IC50 | 8 | — | |
WEKXUMJLGXGLNE
|
8.4 | IC50 | 2 | — | |
LHKFTDVGHHDMKX
|
8.4 | IC50 | 2 | — | |
MNTIFTYMXHJTKW
|
8.4 | IC50 | 2 | — | |
REXKPUWAXOQORC
|
8.4 | IC50 | 2 | — | |
UHTDRCGXSYGMRR
|
8.4 | IC50 | 2 | — | |
SXOAHIZWCZOILH
|
8.4 | IC50 | 3 | — | |
VCYUDKGDSCTDPU
|
8.4 | IC50 | 2 | — | |
VKRFQEVWFMGEEK
|
8.4 | IC50 | 2 | — | |
XRNKNZSYIMJPQE
|
8.4 | IC50 | 2 | — | |
XRNKNZSYIMJPQE
|
8.4 | IC50 | 2 | — | |
AHLGPCZDAPQKRY
|
8.4 | IC50 | 2 | — | |
AOTZMAHOBVGVQU
|
8.4 | IC50 | 3 | — | |
DDOIQOFHDMJGBP
|
8.4 | IC50 | 2 | — | |
UZDFKZMJYSQQHI
|
8.4 | IC50 | 2 | — | |
VBKZDPSLLFEXQC
|
8.4 | IC50 | 2 | — | |
YGLOZPVIZVIBDT
|
8.4 | IC50 | 2 | — | |
AZHGECCHCQEMBR
|
8.4 | IC50 | 2 | — | |
ANUDJEBSNITMOR
|
8.4 | IC50 | 2 | — | |
CYVICQCUAYMJDA
|
8.4 | IC50 | 2 | — | |
FCTMRPTVPHVTTN
|
8.4 | IC50 | 3 | — | |
ICDZOMMZQJGZGT
|
8.4 | IC50 | 2 | — | |
PJGWILKULVRVIE
|
8.4 | IC50 | 2 | — | |
ATFPRZUKXKQMOY
|
8.4 | IC50 | 2 | — | |
OCUQANFWZAMQKA
|
8.4 | IC50 | 2 | — | |
OZRIMKPTCZSADH
|
8.4 | IC50 | 2 | — | |
SQHCXAPOOMTODU
|
8.4 | IC50 | 2 | — | |
YGLOZPVIZVIBDT
|
8.4 | IC50 | 2 | — | |
GULOFVVKGUTUDX
|
8.3 | IC50 | 2 | — | |
HDCONQSFHGFUFZ
|
8.3 | IC50 | 2 | — | |
KQVZYWXQAVPSNP
|
8.3 | IC50 | 2 | — | |
NDHYFBZFYCXQJV
|
8.3 | IC50 | 2 | — | |
YTJUXLJKPMJRBK
|
8.3 | IC50 | 2 | — | |
CAOWMPQVHUJGPS
|
8.3 | IC50 | 2 | — | |
SAECGYZACNUJAE
|
8.3 | IC50 | 2 | — | |
GRFFUKNFLUHFHE
|
8.3 | IC50 | 2 | — | |
QMMKZCBSRMHBGN
|
8.3 | IC50 | 2 | — | |
RJJRKJYXPONNFC
|
8.3 | IC50 | 2 | — | |
AFMUVNRIPITERN
|
8.3 | IC50 | 2 | — | |
APUFQCSYCHYZIW
|
8.3 | IC50 | 2 | — | |
BSGXIJLWDIVEFC
|
8.3 | IC50 | 2 | — | |
DEFPDGLJZGBIGF
|
8.3 | IC50 | 2 | — | |
JHWZVZSMRWIZMO
|
8.3 | IC50 | 2 | — | |
KBNXSZUPQRGYNY
|
8.3 | IC50 | 3 | — | |
CBIUHBBBOUSNQK
|
8.3 | IC50 | 2 | — | |
YKHDDBRKQAIROO
|
8.3 | IC50 | 3 | — | |
DHSOPLGHCCWMQK
|
8.3 | IC50 | 3 | — | |
DVPUCKCSNKRQIM
|
8.3 | IC50 | 2 | — | |
FKPOFESGNHGZMW
|
8.3 | IC50 | 2 | — |