Target Details
| UniProt AC | Q14524 |
|---|---|
| Gene Symbol | SCN5A |
| Protein Name | Sodium channel protein type 5 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 683
- Clinical molecules 2
- Avg pChEMBL 7.49
KEGG Pathways (2)
Associated Diseases (8)
Active Molecules (683)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YUNNMYFFOLAHHL
|
6.1 | IC50 | 2 | — | |
BGEXEHUFMGIZSJ
|
6.1 | IC50 | 2 | — | |
FCGCWVRBOOKMTK
|
6.1 | IC50 | 3 | — | |
GRXUKFHZQDPFAI
|
6.1 | IC50 | 2 | — | |
IJKKZVFOENDHPB
|
6.1 | IC50 | 2 | — | |
MIIOBHGQUATGFU
|
6.1 | IC50 | 2 | — | |
PPKNTGHPZNLOFG
|
6.1 | IC50 | 2 | — | |
WFAAJGGDSHOXSH
|
6.1 | IC50 | 2 | — | |
ZGBOGHHZYOLAIZ
|
6.1 | IC50 | 2 | — | |
NGDMDSQQEVAVIN
|
6.0 | IC50 | 2 | — | |
XJXFPLHCRFQLST
|
6.0 | IC50 | 3 | — | |
IILXZRYSENLMEG
|
6.0 | IC50 | 2 | — | |
HCTZADLXNTVPRR
|
6.0 | IC50 | 2 | — | |
ISRFCSFRFHSLEY
|
6.0 | IC50 | 2 | — | |
JUSUTAPQEPWMEW
|
6.0 | IC50 | 2 | — | |
KFLDDFUYNBKZOT
|
6.0 | IC50 | 2 | — | |
NEGUYMSGZYTTPG
|
6.0 | IC50 | 2 | — | |
TZVKLOBAQHLBCP
|
6.0 | IC50 | 2 | — | |
WVXWILBXLFSUOH
|
6.0 | IC50 | 2 | — | |
AKAQZLFYNGRABJ
|
6.0 | IC50 | 2 | — | |
AVOALNAAWZWOQC
|
6.0 | IC50 | 2 | — | |
LXEBABFPSLDVID
|
6.0 | IC50 | 2 | — | |
NDLBOYOWPCRMAR
|
6.0 | IC50 | 2 | — | |
GUGOEEXESWIERI
|
6.0 | IC50 | 18 | Yes | |
XOKHNIWKPBYBRC
|
6.0 | IC50 | 2 | — | |
ZJRDHGFMVANNGO
|
6.0 | IC50 | 2 | — | |
CFMYXEVWODSLAX
|
6.0 | IC50 | 8 | — | |
FFXBKKBNWGBOAE
|
6.0 | IC50 | 2 | — | |
HZXKYOMFVBZNGK
|
6.0 | IC50 | 2 | — | |
LLCJMXUOUAGOJT
|
6.0 | IC50 | 3 | — | |
RSJUYPGFGAQOLP
|
6.0 | IC50 | 2 | — | |
ULKCBFMHTCGKKY
|
6.0 | IC50 | 2 | — | |
ZBFHVTYUERGXHJ
|
6.0 | IC50 | 2 | — |