Target Details
| UniProt AC | Q14524 |
|---|---|
| Gene Symbol | SCN5A |
| Protein Name | Sodium channel protein type 5 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 683
- Clinical molecules 2
- Avg pChEMBL 7.49
KEGG Pathways (2)
Associated Diseases (8)
Active Molecules (683)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NGDMDSQQEVAVIN
|
6.3 | IC50 | 2 | — | |
SSYPIIPRUWAYCB
|
6.3 | IC50 | 2 | — | |
TVPPCCLUHPATAW
|
6.3 | IC50 | 2 | — | |
UZISDSQSQIPNGM
|
6.3 | IC50 | 2 | — | |
XXQSOIJXIKSRGX
|
6.3 | IC50 | 3 | — | |
FOVUYWGGUYNFBG
|
6.3 | IC50 | 2 | — | |
GKCBAIGFKIBETG
|
6.3 | IC50 | 10 | — | |
RUKSBVHNOBYDMK
|
6.3 | IC50 | 2 | — | |
RIKGAAKYGUUCJR
|
6.3 | IC50 | 2 | — | |
UOTNRDAWNWUHGV
|
6.3 | IC50 | 2 | — | |
JDRAVOBAUSSLSR
|
6.3 | IC50 | 2 | — | |
PPMOJHYERWGAEB
|
6.3 | IC50 | 2 | — | |
SXOAHIZWCZOILH
|
6.3 | IC50 | 9 | — | |
GRLGZDKCJLINRL
|
6.2 | IC50 | 2 | — | |
LYMPFPNZOWWYPE
|
6.2 | IC50 | 2 | — | |
RHNQUMXARXOPCS
|
6.2 | IC50 | 2 | — | |
VSZLPFCJMSEGIJ
|
6.2 | IC50 | 2 | — | |
XVGMRZRHSRQQFG
|
6.2 | IC50 | 2 | — | |
YNUAEEJQYHYLMS
|
6.2 | IC50 | 2 | — | |
WJRHMCNOLMTJKY
|
6.2 | IC50 | 3 | — | |
GNHZBRMVSAIOCC
|
6.2 | IC50 | 2 | — | |
KBOLMQHKSVRFIL
|
6.2 | IC50 | 2 | — | |
KQWOBWMNPNSGDQ
|
6.2 | IC50 | 2 | — | |
OEIJXNGSQJJFRS
|
6.2 | IC50 | 2 | — | |
RQJYQECMAVLMJI
|
6.2 | IC50 | 2 | — | |
UKJAFWJAHPMAKD
|
6.2 | IC50 | 2 | — | |
LLEKPWJKKKVEPI
|
6.2 | IC50 | 2 | — | |
BTKIGPLGDZHMLE
|
6.2 | IC50 | 2 | — | |
GXQQARVXYNJKOH
|
6.2 | IC50 | 2 | — | |
BGTDJFUYZQLYLF
|
6.2 | IC50 | 2 | — | |
IKSUDZQUQOMVKP
|
6.2 | IC50 | 2 | — | |
SHCCRGIIPVJFHB
|
6.2 | IC50 | 2 | — | |
YTFBGOIIROWIRX
|
6.2 | IC50 | 2 | — | |
LEZRONYAEVJQQI
|
6.2 | IC50 | 2 | — | |
YFFAMHITDBOYET
|
6.2 | IC50 | 2 | — | |
MSLIEPIIAJYDTK
|
6.2 | IC50 | 2 | — | |
PDZFTSNLQQQGTI
|
6.2 | IC50 | 2 | — | |
BDPIGJCLXMOTDZ
|
6.1 | IC50 | 2 | — | |
BECROBIDPQYXRW
|
6.1 | IC50 | 2 | — | |
CQNLZLUWQRHCES
|
6.1 | IC50 | 2 | — | |
KTYPXYDRNKHYHU
|
6.1 | IC50 | 2 | — | |
YTSQUJOXQNTPEU
|
6.1 | IC50 | 2 | — | |
ISWVMFZMELKMAQ
|
6.1 | IC50 | 2 | — | |
YYVCJPDYCCNDLJ
|
6.1 | IC50 | 2 | — | |
CZZSYEPBDUZHLQ
|
6.1 | IC50 | 2 | — | |
FYUHLCNXSLHELL
|
6.1 | IC50 | 2 | — | |
XSDQTOBWRPYKKA
|
6.1 | IC50 | 2 | — | |
ZGBCYVXZLVHZHE
|
6.1 | IC50 | 2 | — | |
DFBDAHMZXJYZJG
|
6.1 | IC50 | 7 | — | |
UXBLZIZAOQSOGB
|
6.1 | IC50 | 2 | — |