Target Details
| UniProt AC | Q14524 |
|---|---|
| Gene Symbol | SCN5A |
| Protein Name | Sodium channel protein type 5 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 683
- Clinical molecules 2
- Avg pChEMBL 7.49
KEGG Pathways (2)
Associated Diseases (8)
Active Molecules (683)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JFTTWRHSUYMBCX
|
6.5 | IC50 | 2 | — | |
WXZNLCQMGILZDR
|
6.5 | IC50 | 2 | — | |
QOBHARXOODMEIE
|
6.5 | IC50 | 2 | — | |
RVFFHAQSQFHDKW
|
6.5 | IC50 | 2 | — | |
UTAOYMGDFRTJNO
|
6.5 | IC50 | 2 | — | |
DWIFDJBIHHABLE
|
6.5 | IC50 | 2 | — | |
FNDAXQFHRLFJSB
|
6.5 | IC50 | 2 | — | |
ODMZUCMOJODESH
|
6.5 | IC50 | 2 | — | |
FEVBKJITJDHASC
|
6.5 | IC50 | 3 | — | |
QWEHIZAOKREMOE
|
6.5 | IC50 | 2 | — | |
BHJSCRNVDBKWGW
|
6.5 | IC50 | 2 | — | |
CVHPNFWHLXBWPR
|
6.5 | IC50 | 2 | — | |
DLJIYRWMNZPEPW
|
6.5 | IC50 | 2 | — | |
IXPTYEXVNBRWNJ
|
6.5 | IC50 | 2 | — | |
JKJROAPYAHIAJY
|
6.5 | IC50 | 2 | — | |
NESLCFXDKPAXII
|
6.5 | IC50 | 2 | — | |
LIJVHEHWJNGQJH
|
6.4 | IC50 | 2 | — | |
AFULOBBVYHAEMW
|
6.4 | IC50 | 2 | — | |
JYYKEMPXQHPLKT
|
6.4 | IC50 | 3 | — | |
NXOLRSKOGVZGJE
|
6.4 | IC50 | 2 | — | |
QNQNMXVCAYGWFY
|
6.4 | IC50 | 2 | — | |
RGEBGRLYAPVJLZ
|
6.4 | IC50 | 2 | — | |
UKJAFWJAHPMAKD
|
6.4 | IC50 | 2 | — | |
UTAOYMGDFRTJNO
|
6.4 | IC50 | 2 | — | |
UTICZDOENGIDOA
|
6.4 | IC50 | 2 | — | |
VUCGOPZDZHFBHO
|
6.4 | IC50 | 2 | — | |
IFRGFTQIIMWCJG
|
6.4 | IC50 | 2 | — | |
ISNMDOLXNFQPJG
|
6.4 | IC50 | 2 | — | |
SDOGULGNBMMVTH
|
6.4 | IC50 | 2 | — | |
WRIZTMCLCILPFZ
|
6.4 | IC50 | 2 | — | |
WVDCPYJACILIGO
|
6.4 | IC50 | 2 | — | |
YCLDIBUXJUIEOU
|
6.4 | IC50 | 2 | — | |
CSGMIVCOTWOCPC
|
6.3 | IC50 | 2 | — | |
IVNAEBIOSDTKSX
|
6.3 | IC50 | 2 | — | |
KQQXPTRMUYKUIC
|
6.3 | IC50 | 8 | — | |
WVDCPYJACILIGO
|
6.3 | IC50 | 2 | — | |
JHTBXYQIHWCGPI
|
6.3 | IC50 | 2 | — | |
ODIAQAJCRITKNJ
|
6.3 | IC50 | 2 | — | |
PMMALHFQLZXMOO
|
6.3 | IC50 | 2 | — | |
IXDCXFJUPLJBMC
|
6.3 | IC50 | 2 | — | |
RRCQMMXZKUITON
|
6.3 | IC50 | 2 | — | |
NSUPANGHWGJPCM
|
6.3 | IC50 | 2 | — | |
ZMOPTLXEYOVARP
|
6.3 | IC50 | 14 | Yes | |
DTWJNQKJWMKSFE
|
6.3 | IC50 | 2 | — | |
HDIMCCGWDRZXNB
|
6.3 | IC50 | 2 | — | |
QMVCLINXNJGGFP
|
6.3 | IC50 | 2 | — | |
BEBRFALPYNNCLU
|
6.3 | IC50 | 2 | — | |
HBNPJJILLOYFJU
|
6.3 | IC50 | 21 | — | |
JEEZZJOSUGMGIG
|
6.3 | IC50 | 2 | — | |
MOGUMJAJYFSRJV
|
6.3 | IC50 | 3 | — |