Target Details
| UniProt AC | Q14524 |
|---|---|
| Gene Symbol | SCN5A |
| Protein Name | Sodium channel protein type 5 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 683
- Clinical molecules 2
- Avg pChEMBL 7.49
KEGG Pathways (2)
Associated Diseases (8)
Active Molecules (683)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NEBUOXBYNAHKFV
|
7.1 | IC50 | 5 | — | |
VENWKQHIOIEAII
|
7.1 | IC50 | 3 | — | |
OFMOIJVBLHFGHB
|
7.0 | IC50 | 2 | — | |
WOOZKYJTHJWUFV
|
7.0 | IC50 | 2 | — | |
XKWUOIWEHZPVIB
|
7.0 | IC50 | 2 | — | |
XOAUGYVLRSCGBG
|
7.0 | IC50 | 8 | — | |
ALXYLFDRNLWAJQ
|
7.0 | IC50 | 2 | — | |
DHFLDZDCXCPNAT
|
7.0 | IC50 | 2 | — | |
MWDXQRJBADDXCQ
|
7.0 | IC50 | 2 | — | |
QZPUVBFHUUQSFZ
|
7.0 | IC50 | 2 | — | |
ZLWJSZSVEMPEKG
|
7.0 | IC50 | 2 | — | |
AADZPNRBAZVGNN
|
7.0 | IC50 | 2 | — | |
HJTNQQWICWEECK
|
7.0 | IC50 | 3 | — | |
LLQGWDGJRDPIES
|
7.0 | IC50 | 2 | — | |
MCBCKBHAGLJKPH
|
7.0 | IC50 | 2 | — | |
OETZKAGCLMZSKS
|
7.0 | IC50 | 2 | — | |
WDENVSHHVGKVLV
|
7.0 | IC50 | 2 | — | |
OZAYOHJGXLWETR
|
7.0 | IC50 | 2 | — | |
APNKIFBEFRZJNR
|
7.0 | IC50 | 2 | — | |
FPERPEQIXLOVIK
|
7.0 | IC50 | 5 | — | |
IMUKSSQOUCDNFP
|
7.0 | IC50 | 2 | — | |
JZGNUJUVVQHLMQ
|
7.0 | IC50 | 2 | — | |
YJDICZSISKZEKO
|
7.0 | IC50 | 2 | — | |
IMNAMBYRWSGKHX
|
7.0 | IC50 | 3 | — | |
GCKAUEWKJKBEPC
|
6.9 | IC50 | 2 | — | |
RCPKTZHXPBTTTM
|
6.9 | IC50 | 2 | — | |
AKEOVDDAHTWBGN
|
6.9 | IC50 | 3 | — | |
OEHODXUDKGXIAC
|
6.9 | IC50 | 2 | — | |
UMLBPTKZCLVUIO
|
6.9 | IC50 | 2 | — | |
WPCMGHHEOJLHRM
|
6.9 | IC50 | 2 | — | |
NIUMYXYWSPDBFW
|
6.9 | IC50 | 2 | — | |
CXCZBWCPIJUCFH
|
6.9 | IC50 | 2 | — | |
ADMLHCZRKYFTCM
|
6.9 | IC50 | 2 | — | |
UNPJOXGIHJVJQC
|
6.9 | IC50 | 2 | — | |
WTQGKPCUKPVRSK
|
6.9 | IC50 | 2 | — | |
IRKLGNYNAXCIJW
|
6.9 | IC50 | 2 | — | |
ACVOHQCMVBHBMM
|
6.9 | IC50 | 2 | — | |
DSSSTXWTCIBGSG
|
6.8 | IC50 | 2 | — | |
GQJOVRAJLZZUTH
|
6.8 | IC50 | 2 | — | |
NJKBBVDDLCQVAF
|
6.8 | IC50 | 2 | — | |
QBWNJYLTWMVCJV
|
6.8 | IC50 | 2 | — | |
JDJPOKWOABXJKL
|
6.8 | IC50 | 2 | — | |
LNSGKRRBOFFWLA
|
6.8 | IC50 | 2 | — | |
TZUOZTCIJCIQGB
|
6.8 | IC50 | 3 | — | |
DKYUUKRMMHLYCZ
|
6.8 | IC50 | 2 | — | |
FQHDBBOTIYOYLF
|
6.8 | IC50 | 3 | — | |
GAUCTMQMNSDYNT
|
6.8 | IC50 | 2 | — | |
KDOYGXBJAYKYQW
|
6.8 | IC50 | 2 | — | |
PWIGOAGIFOIPHV
|
6.8 | IC50 | 2 | — | |
RFZHHXIXCJHZNR
|
6.8 | IC50 | 2 | — |