Target Details
| UniProt AC | Q14416 |
|---|---|
| Gene Symbol | GRM2 |
| Protein Name | Metabotropic glutamate receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00003 (7tm_3) PF01094 (ANF_receptor) PF07562 (NCD3G) |
Summary
- Multi-target molecules 134
- Clinical molecules 0
- Avg pChEMBL 7.1
KEGG Pathways (5)
Active Molecules (134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
INNYBEXRWKVEPM
|
6.6 | Ki | 2 | — | |
KEOUMVRTMMZTEV
|
6.6 | IC50 | 2 | — | |
XMENKXPGVGTNAZ
|
6.6 | Ki | 2 | — | |
ASNFTDCKZKHJSW
|
6.6 | Ki | 5 | — | |
CNBSEOHDTNDGOV
|
6.5 | IC50 | 2 | — | |
ZDVZEEBBIZFFGQ
|
6.5 | Ki | 2 | — | |
JJWWDQCTTPDNGK
|
6.5 | IC50 | 2 | — | |
KPKSEPNXKJWVTO
|
6.5 | IC50 | 2 | — | |
NEVQUXDVNDJANK
|
6.5 | Ki | 2 | — | |
JCGJEPFYMOHIDP
|
6.5 | Ki | 2 | — | |
YLOYRSFMNLQTKN
|
6.5 | Ki | 2 | — | |
INNYBEXRWKVEPM
|
6.5 | Ki | 2 | — | |
JYWMNSYAIWOJGC
|
6.5 | IC50 | 2 | — | |
RNGJMJZHZIDZHG
|
6.4 | Ki | 2 | — | |
SGCNJDYPITVHEN
|
6.4 | IC50 | 2 | — | |
BQVZICWQBFTOJX
|
6.4 | Ki | 2 | — | |
QMTVYANBFIIHRR
|
6.4 | Ki | 2 | — | |
UCGGDVUKMWZJLA
|
6.4 | IC50 | 2 | — | |
UXNRHIJPZNNDDJ
|
6.4 | Ki | 2 | — | |
IRMXEKLCWFUGDP
|
6.4 | IC50 | 2 | — | |
XZFMJVJDSYRWDQ
|
6.3 | Ki | 2 | — | |
GZOVEPYOCJWRFC
|
6.3 | Ki | 2 | — | |
MHGNPCZGYOTMGN
|
6.2 | Ki | 2 | — | |
AQCRJOWGCAFEAA
|
6.2 | Ki | 2 | — | |
BQVZICWQBFTOJX
|
6.2 | Ki | 2 | — | |
DDOQBQRIEWHWBT
|
6.2 | Ki | 4 | — | |
YQHUAECMPKPVHE
|
6.1 | Ki | 2 | — | |
SLBQKYUURZKYBP
|
6.1 | Ki | 2 | — | |
RKBRDSPEJMNTGE
|
6.1 | IC50 | 2 | — | |
APZIMAYYQKOWFP
|
6.0 | Ki | 2 | — | |
XMDHIHAVEVYYTH
|
6.0 | Ki | 2 | — | |
UBOUWUOIJSJJIT
|
6.0 | IC50 | 2 | — | |
XAWBHQAHNLHFPV
|
6.0 | IC50 | 2 | — | |
ZLLVGXOCXYGTFK
|
6.0 | IC50 | 2 | — |