Target Details
| UniProt AC | Q14416 |
|---|---|
| Gene Symbol | GRM2 |
| Protein Name | Metabotropic glutamate receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00003 (7tm_3) PF01094 (ANF_receptor) PF07562 (NCD3G) |
Summary
- Multi-target molecules 134
- Clinical molecules 0
- Avg pChEMBL 7.1
KEGG Pathways (5)
Active Molecules (134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LETPPZNSGLCXSE
|
9.0 | Ki | 3 | — | |
YASVRZWVUGJELU
|
8.6 | Ki | 3 | — | |
QBHIOYZCUZBIEN
|
8.4 | Ki | 2 | — | |
PYCDNJSXQRXRFH
|
8.4 | Ki | 2 | — | |
GZOVEPYOCJWRFC
|
8.3 | Ki | 2 | — | |
PVCLSZDVATUGHR
|
8.3 | IC50 | 2 | — | |
VHWZAFAIQMVWBH
|
8.3 | IC50 | 2 | — | |
BLUDMDWTHRXJRA
|
8.2 | IC50 | 2 | — | |
ALTAMTJSSZBUFX
|
8.2 | IC50 | 2 | — | |
ZYGZDPKEZBLAHD
|
8.2 | IC50 | 2 | — | |
LFAGGDAZZKUVKO
|
8.2 | IC50 | 2 | — | |
HHUBIRLCPJRLDB
|
8.1 | Ki | 2 | — | |
PCFAQNCKPHVYDF
|
8.0 | IC50 | 2 | — | |
QHBLXVIRCXAIGL
|
8.0 | IC50 | 2 | — | |
DWHFXDLHZUPSDA
|
7.9 | IC50 | 2 | — | |
XBQXBDVFZNVFIQ
|
7.9 | IC50 | 2 | — | |
HQTAUDRHEUIJTC
|
7.9 | Ki | 2 | — | |
YASVRZWVUGJELU
|
7.8 | Ki | 3 | — | |
VBZWVJXSTPCEIR
|
7.8 | IC50 | 2 | — | |
BQAVZGJJQFJSMW
|
7.8 | IC50 | 2 | — | |
UYDTVURQQQIWQU
|
7.8 | IC50 | 2 | — | |
AAQAEWBPCIXLCR
|
7.8 | IC50 | 2 | — | |
XJEBSHOFIMSIIB
|
7.8 | IC50 | 2 | — | |
FUOXGTLPOUSBMV
|
7.7 | IC50 | 2 | — | |
WSIUIRJCBSRFHV
|
7.7 | IC50 | 2 | — | |
OCNVADMKXAQCFP
|
7.7 | IC50 | 2 | — | |
IJUVTLSGLODULR
|
7.7 | IC50 | 2 | — | |
PSQSAQVJYBYDHR
|
7.7 | IC50 | 2 | — | |
VLZBRVJVCCNPRJ
|
7.7 | IC50 | 4 | — | |
QSNQXCLTDBTOIU
|
7.7 | IC50 | 2 | — | |
LGSORWLWDBCUMM
|
7.6 | Ki | 2 | — | |
LVVJEBBNZXFVDH
|
7.6 | IC50 | 2 | — | |
CVAFGISXRYNCDR
|
7.6 | IC50 | 2 | — | |
ACVCREFNDLDKHC
|
7.6 | IC50 | 2 | — | |
CETJSTBZOJQTPJ
|
7.6 | IC50 | 2 | — | |
PZICKINIOPPAGP
|
7.6 | Ki | 2 | — | |
YKPDUULXXDPIGO
|
7.6 | IC50 | 2 | — | |
XEAYLXSKXSSPLU
|
7.5 | IC50 | 2 | — | |
OKBTYHHXUOFYFO
|
7.5 | IC50 | 2 | — | |
WNOZOUHFGZKGNT
|
7.5 | IC50 | 2 | — | |
DPFFCWQLYRMZOU
|
7.5 | Ki | 2 | — | |
OSPUMEGCPJZZKB
|
7.5 | IC50 | 2 | — | |
ZGEPFYVQFLRUIH
|
7.5 | IC50 | 2 | — | |
NZZMAEBSZGFPBU
|
7.5 | IC50 | 2 | — | |
UFMGYRJFXQXVOH
|
7.4 | IC50 | 2 | — | |
XLSMUHMCZSVHHK
|
7.4 | IC50 | 2 | — | |
XMDLTKGXRPVDSY
|
7.4 | IC50 | 2 | — | |
UOCRQSAPAFCFKX
|
7.3 | IC50 | 2 | — | |
XMENKXPGVGTNAZ
|
7.3 | IC50 | 2 | — | |
UVWURBJBVZRMKJ
|
7.3 | Ki | 2 | — |