Target Details
| UniProt AC | Q14397 |
|---|---|
| Gene Symbol | GCKR |
| Protein Name | Glucokinase regulatory protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF20741 (GKRP-like_C) PF22198 (GKRP_SIS_2) PF22645 (GKRP_SIS_N) |
Summary
- Multi-target molecules 32
- Clinical molecules 0
- Avg pChEMBL 7.07
Top Co-occurrence Targets
- GCK 32 shared
Active Molecules (32)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NVRHWELRHNYZOU
|
8.2 | IC50 | 2 | — | |
LJCXNEAHAINFGA
|
8.2 | IC50 | 2 | — | |
NVRHWELRHNYZOU
|
8.0 | IC50 | 2 | — | |
PKUYDBKKSMGBJL
|
7.8 | IC50 | 2 | — | |
QBAPAHDQINABPY
|
7.8 | IC50 | 2 | — | |
UEFBMKGVQXOXRD
|
7.8 | IC50 | 2 | — | |
SZCHUQJVAMEDBM
|
7.7 | IC50 | 2 | — | |
UEFBMKGVQXOXRD
|
7.6 | IC50 | 2 | — | |
UEFBMKGVQXOXRD
|
7.4 | IC50 | 2 | — | |
UMAJLFWMSYDGBK
|
7.4 | IC50 | 2 | — | |
BXXBQXYOMZHUMV
|
7.4 | IC50 | 2 | — | |
WNQFIUIJXPOGMC
|
7.3 | IC50 | 2 | — | |
NVRHWELRHNYZOU
|
7.2 | IC50 | 2 | — | |
QDURMADQEYTVDK
|
7.2 | IC50 | 2 | — | |
WKJNWGUQBRFMBN
|
7.1 | IC50 | 2 | — | |
KYAOTPJIJKJOOX
|
7.0 | IC50 | 2 | — | |
IBDJORYQEKQDSY
|
7.0 | IC50 | 2 | — | |
AYCYQFOAZRLEHT
|
6.9 | IC50 | 2 | — | |
KMKJDWRQGUEOJR
|
6.9 | IC50 | 2 | — | |
UENQSWPRHPUNQA
|
6.8 | IC50 | 2 | — | |
ZNYWQWSQKLMSTM
|
6.8 | IC50 | 2 | — | |
RCCQDYKCTOZGFC
|
6.7 | IC50 | 2 | — | |
NINQGEYFRYPZAJ
|
6.6 | IC50 | 2 | — | |
PXOBWRSOEJFIBJ
|
6.6 | IC50 | 2 | — | |
WRPSYMIONPCVAD
|
6.6 | IC50 | 2 | — | |
KQUYOJWMGJXOCW
|
6.5 | IC50 | 2 | — | |
OWHJVXHDOFJZEK
|
6.5 | IC50 | 2 | — | |
OLLSTZGMQOPNQB
|
6.4 | IC50 | 2 | — | |
CNCSRJXQZGFKQH
|
6.3 | IC50 | 2 | — | |
VEMNCZMADJQYTF
|
6.3 | IC50 | 2 | — | |
VBDHWHUISVHCNK
|
6.1 | IC50 | 2 | — | |
XOWBHNIRCZERRH
|
6.0 | IC50 | 2 | — |