Target Details
| UniProt AC | Q14289 |
|---|---|
| Gene Symbol | PTK2B |
| Protein Name | Protein-tyrosine kinase 2-beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21477 (FERM_C_FAK1) PF00373 (FERM_M) PF18038 (FERM_N_2) PF03623 (Focal_AT) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 210
- Clinical molecules 15
- Avg pChEMBL 7.28
KEGG Pathways (11)
- Cadherin signaling
- Calcium signaling pathway
- Chemokine signaling pathway
- GnRH signaling pathway
- Hepatitis B
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Leukocyte transendothelial migration
- Natural killer cell mediated cytotoxicity
- Phospholipase D signaling pathway
- Yersinia infection
Active Molecules (210)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MHCPAORAYMTGCZ
|
6.0 | Ki | 37 | — | |
MQRDVGBWWVWMEN
|
6.0 | Ki | 47 | — | |
MVCOAUNKQVWQHZ
|
6.0 | Kd | 54 | Yes | |
OWDRQHVEJIYVOI
|
6.0 | Ki | 47 | — | |
SJMCNVUMRNUOKS
|
6.0 | IC50 | 2 | — | |
STISJUSFFZAZMP
|
6.0 | Ki | 7 | — | |
UQRCJCNVNUFYDX
|
6.0 | Kd | 27 | — | |
XOVPCPRZRHQFBI
|
6.0 | Ki | 15 | — |