Target Details
| UniProt AC | Q14289 |
|---|---|
| Gene Symbol | PTK2B |
| Protein Name | Protein-tyrosine kinase 2-beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21477 (FERM_C_FAK1) PF00373 (FERM_M) PF18038 (FERM_N_2) PF03623 (Focal_AT) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 210
- Clinical molecules 15
- Avg pChEMBL 7.28
KEGG Pathways (11)
- Cadherin signaling
- Calcium signaling pathway
- Chemokine signaling pathway
- GnRH signaling pathway
- Hepatitis B
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Leukocyte transendothelial migration
- Natural killer cell mediated cytotoxicity
- Phospholipase D signaling pathway
- Yersinia infection
Active Molecules (210)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FBCYLDMQAGIHQR
|
6.6 | Kd | 2 | — | |
GCYXEGSPUDSZJY
|
6.6 | Ki | 82 | — | |
HESLKTSGTIBHJU
|
6.6 | Kd | 6 | — | |
LRZYYIZFBXFSJB
|
6.6 | Ki | 69 | — | |
MCCCQFAOMZMZKE
|
6.6 | Ki | 52 | — | |
VKBFHTIUXUCYRQ
|
6.6 | Ki | 66 | — | |
RVULLEYKHMQYRU
|
6.6 | IC50 | 2 | — | |
RYYNGWLOYLRZLK
|
6.6 | Kd | 45 | — | |
MGGBYMDAPCCKCT
|
6.6 | Kd | 23 | — | |
NMJMRSQTDLRCRQ
|
6.5 | IC50 | 7 | — | |
GNOZTUOADYKOFQ
|
6.5 | IC50 | 5 | — | |
PHXJVRSECIGDHY
|
6.5 | Kd | 59 | — | |
XQVVPGYIWAGRNI
|
6.5 | Kd | 34 | — | |
HEUSUIRCBWROMH
|
6.5 | Ki | 64 | — | |
WUWDLXZGHZSWQZ
|
6.5 | Ki | 41 | — | |
NSKYYUZMAXEZIR
|
6.5 | Ki | 15 | — | |
LCVIRAZGMYMNNT
|
6.5 | Kd | 20 | — | |
CFIBXVQLBVNOHW
|
6.4 | Ki | 64 | — | |
XJSFDMGICAWQFS
|
6.4 | Ki | 60 | — | |
INQBVHWEOAKYED
|
6.4 | IC50 | 2 | — | |
BIKYDWLMTPRSQL
|
6.3 | Ki | 50 | — | |
GDYZFFBMSBDTAA
|
6.3 | Ki | 60 | — | |
JAMDNXUAYUHJLJ
|
6.3 | Ki | 40 | — | |
NJPWCTYVEJIQBM
|
6.3 | Ki | 72 | — | |
PCQMERRARZKTPW
|
6.3 | Ki | 68 | — | |
XHORJSJFHVABEA
|
6.3 | Ki | 49 | — | |
ODPGGGTTYSGTGO
|
6.3 | Kd | 153 | — | |
IGFFFJZWKLOHRI
|
6.2 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
6.2 | Kd | 151 | — | |
IAYGCINLNONXHY
|
6.2 | Kd | 50 | — | |
OPWPQZXQSROBLU
|
6.2 | IC50 | 2 | — | |
PSCJSWRVCKUMSL
|
6.2 | Ki | 35 | — | |
RJZDECGDCKOHBV
|
6.2 | Ki | 70 | — | |
XQVVPGYIWAGRNI
|
6.2 | Ki | 19 | — | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 91 | Yes | |
DAJMEJBPGNBYEH
|
6.2 | IC50 | 2 | — | |
BJRRXLJCIAUKMM
|
6.1 | IC50 | 2 | — | |
GUBJNPWVIUFSTR
|
6.1 | Kd | 103 | — | |
YYLKKYCXAOBSRM
|
6.1 | Kd | 191 | — | |
CHTMRWQLNNRRFJ
|
6.1 | Ki | 70 | — | |
MTCHQDWUHQADSY
|
6.1 | Ki | 29 | — | |
VXYDJXMHISGSDA
|
6.1 | Ki | 59 | — | |
YUOWJICKAJQZLS
|
6.1 | Ki | 35 | — | |
OYONTEXKYJZFHA
|
6.0 | Kd | 69 | Yes | |
WVMANZPBOBRWCB
|
6.0 | Ki | 9 | — | |
BPNUQXPIQBZCMR
|
6.0 | Ki | 60 | — | |
IJNGXROUMFEKDB
|
6.0 | Ki | 39 | — | |
IOBVCHJTLVPPBR
|
6.0 | Ki | 39 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |