Target Details
| UniProt AC | Q14289 |
|---|---|
| Gene Symbol | PTK2B |
| Protein Name | Protein-tyrosine kinase 2-beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21477 (FERM_C_FAK1) PF00373 (FERM_M) PF18038 (FERM_N_2) PF03623 (Focal_AT) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 210
- Clinical molecules 15
- Avg pChEMBL 7.28
KEGG Pathways (11)
- Cadherin signaling
- Calcium signaling pathway
- Chemokine signaling pathway
- GnRH signaling pathway
- Hepatitis B
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Leukocyte transendothelial migration
- Natural killer cell mediated cytotoxicity
- Phospholipase D signaling pathway
- Yersinia infection
Active Molecules (210)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OEVBGOMMLVZIHM
|
7.3 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.3 | Kd | 64 | Yes | |
QGXMVFJEJZPAES
|
7.3 | Ki | 2 | — | |
IAHRSPNDVKURFK
|
7.3 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
7.2 | Kd | 200 | — | |
OKUZSDKSFUEYGG
|
7.2 | Ki | 2 | — | |
QQXRXXYLRNDAPS
|
7.2 | Ki | 2 | — | |
XOOAAYRIVATZNM
|
7.2 | Ki | 55 | — | |
BBZHHJCMVZXOQN
|
7.2 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
7.1 | Kd | 170 | — | |
XTLUDGUIOTYGQW
|
7.1 | Ki | 2 | — | |
HZTYDQRUAWIZRE
|
7.1 | Kd | 40 | Yes | |
WINHZLLDWRZWRT
|
7.1 | Kd | 201 | Yes | |
XZXHXSATPCNXJR
|
7.1 | Kd | 165 | Yes | |
MUVVMGFRHXQCRG
|
7.1 | Ki | 2 | — | |
QGXMVFJEJZPAES
|
7.1 | Ki | 2 | — | |
FWLMVFUGMHIOAA
|
7.1 | IC50 | 26 | — | |
CXQHYVUVSFXTMY
|
7.0 | Kd | 154 | — | |
DBXGGXLBTWZXBB
|
7.0 | Ki | 39 | — | |
ZVWRFVCNQOECJS
|
7.0 | Ki | 71 | — | |
XHUZMLCGFNWCHH
|
7.0 | Ki | 2 | — | |
CAHNFGYWMWNXMR
|
6.9 | IC50 | 9 | — | |
YHVHYWYQEFELOW
|
6.9 | IC50 | 44 | — | |
ALKJNCZNEOTEMP
|
6.9 | Kd | 55 | — | |
SVXALMKNVZGHQH
|
6.9 | IC50 | 2 | — | |
AZSAXICINIVCFK
|
6.9 | IC50 | 2 | — | |
PTVPBWWDGZSEAF
|
6.9 | Ki | 63 | — | |
WINHZLLDWRZWRT
|
6.9 | Ki | 66 | — | |
HIHOEGPXVVKJPP
|
6.9 | IC50 | 10 | — | |
JISGJXUNHIZAJK
|
6.9 | Ki | 2 | — | |
HZHMSBKFDZWRLC
|
6.8 | IC50 | 2 | — | |
OHGGKMIGVXXLRP
|
6.8 | Ki | 2 | — | |
JSKUWFIZUALZLX
|
6.8 | Ki | 33 | — | |
KTEIFNKAUNYNJU
|
6.8 | Ki | 48 | — | |
QHPODLYCTXKTMR
|
6.8 | Ki | 2 | — | |
JPEPNPZDXMQVKW
|
6.8 | Ki | 2 | — | |
LQVXSNNAFNGRAH
|
6.8 | Kd | 33 | Yes | |
WVXNSAVVKYZVOE
|
6.8 | IC50 | 92 | — | |
ZCCPLJOKGAACRT
|
6.8 | Kd | 599 | — | |
PLNNDRULHJUPFM
|
6.7 | Ki | 2 | — | |
KTEIFNKAUNYNJU
|
6.7 | Kd | 114 | — | |
NZNRLSKYWIKFMQ
|
6.7 | IC50 | 3 | — | |
PBCZSGKMGDDXIJ
|
6.7 | Kd | 68 | Yes | |
WKDACQVEJIVHMZ
|
6.7 | Kd | 46 | — | |
PUPCRRRSBUYJAD
|
6.7 | Ki | 44 | Yes | |
RTDSHUGNRVXRHN
|
6.7 | Ki | 51 | — | |
XHVOZHLINNPOHR
|
6.7 | IC50 | 2 | — | |
HJHMZOIXHWLHQD
|
6.7 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
6.7 | Kd | 139 | — | |
UBPYILGKFZZVDX
|
6.6 | IC50 | 130 | Yes |